SCHEMBL4392079

SCHEMBL4392079

[CH2]CNc1nc(NCc2ccc(Cl)cc2)ncc1N

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 2/20 0.46
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
PRKCQ Q04759 2/20 0.44
APP P05067 2/20 0.44
NTRK1 P04629 1/20 0.42
IGF1R P08069 1/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAP4K4 O95819 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4386385 0.84 HDAC3 (0.51) HDAC3HDAC1HDAC2HDAC6NTRK1
SCHEMBL4394654 0.84 APP (0.49) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL4392092 0.82 RPS6KB1 (0.43) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL4387694 0.82 DYRK1A (0.41) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL10996739 0.79 VNN1 (0.51) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL3186194 0.79 VNN1 (0.46) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL4387931 0.78 PRKCQ (0.67) PRKCQALDH1A1MAP4K4PKM
SCHEMBL4385162 0.76 NTRK1 (0.49) PRKCQAPPNTRK1
SCHEMBL21436684 0.70 APP (0.49) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL9681910 0.70 APP (0.47) VNN1HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2131844-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV Therapeutics Inc. (US) 2009-12-16 EP disclosed
WO-2008123891-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV THERAPEUTICS, INC. (US) 2008-10-16 WO disclosed