SCHEMBL4385162

SCHEMBL4385162

[CH2]CNc1nc(NCc2cccc(F)c2)ncc1N

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 12/20 0.49
APP P05067 2/20 0.49
PRKCQ Q04759 1/20 0.48
CCNT1 O60563 1/20 0.45
RPS6KB1 P23443 1/20 0.44
JAK2 O60674 1/20 0.43
JAK1 P23458 1/20 0.43
JAK3 P52333 1/20 0.43
PLK4 O00444 1/20 0.43
PAK4 O96013 1/20 0.43
PTK2 Q05397 1/20 0.42
NTRK3 Q16288 1/20 0.42
NTRK2 Q16620 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4394654 0.85 APP (0.49) APPPRKCQRPS6KB1JAK2JAK1
SCHEMBL4392092 0.83 RPS6KB1 (0.43) NTRK1RPS6KB1PLK4
SCHEMBL3192248 0.81 NTRK1 (0.48) NTRK1APPPRKCQRPS6KB1JAK2
SCHEMBL4386385 0.80 HDAC3 (0.51) NTRK1
SCHEMBL4387694 0.80 DYRK1A (0.41) NTRK1PRKCQRPS6KB1
SCHEMBL4380044 0.80 PRKCQ (0.69) NTRK1PRKCQ
SCHEMBL4392079 0.76 VNN1 (0.46) NTRK1APPPRKCQ
SCHEMBL26429360 0.74 APP (0.54) NTRK1APPPRKCQCCNT1RPS6KB1
SCHEMBL22191429 0.73 GAA (0.52) NTRK1APPPRKCQCCNT1RPS6KB1
SCHEMBL25934296 0.72 GAA (0.51) NTRK1APPPRKCQCCNT1RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2131844-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV Therapeutics Inc. (US) 2009-12-16 EP disclosed
WO-2008123891-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV THERAPEUTICS, INC. (US) 2008-10-16 WO disclosed