SCHEMBL4392092

SCHEMBL4392092

[CH2]CNc1nc(NCc2ccc(F)c(F)c2)ncc1N

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 2/20 0.43
VNN1 O95497 4/20 0.42
PLK4 O00444 1/20 0.41
NTRK1 P04629 2/20 0.39
AURKA O14965 1/20 0.38
PIM1 P11309 1/20 0.38
GPR68 Q15743 1/20 0.38
DYRK1A Q13627 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
BCDIN3D Q7Z5W3 1/20 0.35
PDPK1 O15530 2/20 0.35
ABL1 P00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4386385 0.89 HDAC3 (0.51) NTRK1DYRK1ACLK4HDAC3HDAC1
SCHEMBL4387694 0.89 DYRK1A (0.41) RPS6KB1NTRK1DYRK1ACLK4HDAC3
SCHEMBL4385162 0.83 NTRK1 (0.49) RPS6KB1PLK4NTRK1
SCHEMBL4392079 0.82 VNN1 (0.46) VNN1NTRK1HDAC3HDAC1HDAC2
SCHEMBL4394654 0.81 APP (0.49) RPS6KB1VNN1HDAC3HDAC1HDAC2
SCHEMBL3191032 0.81 VNN1 (0.43) RPS6KB1VNN1PLK4AURKAHDAC3
SCHEMBL4384306 0.79 PRKCQ (0.53)
SCHEMBL3192454 0.71 HDAC3 (0.41) NTRK1HDAC3HDAC1HDAC2HDAC6
SCHEMBL3189750 0.71 HDAC3 (0.51) NTRK1HDAC3HDAC1HDAC2HDAC6
SCHEMBL12185810 0.70 LMNA (0.45) AURKAHDAC1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2131844-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV Therapeutics Inc. (US) 2009-12-16 EP disclosed
WO-2008123891-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV THERAPEUTICS, INC. (US) 2008-10-16 WO disclosed