SCHEMBL4392467

SCHEMBL4392467

COC(=O)Oc1cc(OC(=O)OC)c(-c2cccc(OC)c2)c(C(C(C)=O)C(=O)OC)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
ADORA3 P0DMS8 2/20 0.38
ADORA2B P29275 2/20 0.38
ADORA1 P30542 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ADORA2A P29274 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MTNR1A P48039 9/20 0.37
MTNR1B P49286 9/20 0.37
FPR1 P21462 1/20 0.36
HSD17B2 P37059 1/20 0.36
ERN1 O75460 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4385956 0.89 KDM4E (0.40) ADORA3KDM4EALDH1A1HPGDRAB9A
SCHEMBL4381894 0.83 MTNR1A (0.42) HSP90AA1HSP90AB1KDM4EALDH1A1HPGD
SCHEMBL4380826 0.82 CAPN1 (0.38) HSP90AA1HSP90AB1NPC1ALDH1A1RAB9A
SCHEMBL4391759 0.78 HDAC4 (0.43) HSP90AA1HSP90AB1ADORA3ADORA2BADORA1
SCHEMBL4380779 0.70 TDP1 (0.42) KDM4ENPC1ALDH1A1HPGDRAB9A
SCHEMBL4388446 0.70 EGFR (0.40) RAB9A
SCHEMBL6312058 0.70 MTNR1A (0.51) NPC1ALDH1A1RAB9AMTNR1AMTNR1B
SCHEMBL19320327 0.69 RXRA (0.51) ADORA3ADORA2BADORA1
SCHEMBL13135118 0.69 MTNR1B (0.57) NPC1RAB9AMTNR1AMTNR1B
SCHEMBL4392454 0.68 ADORA3 (0.40) HSP90AA1HSP90AB1ADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7538241-B2 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-05-26 US disclosed
US-20070155813-A1 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-07-05 US disclosed
EP-1704856-A1 HSP90 FAMILY PROTEIN INHIBITOR KYOWA HAKKO KOGYO CO., LTD. (JP) 2006-09-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070155813-A1 Hsp90 family protein inhibitors HSP90AB1, HEATR1, HSP90AB2P HSP90AA1 5/4885HSP90AB1 1/4885ADORA3 3728/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.