SCHEMBL43927

SCHEMBL43927

O=C(CI)Nc1ccc(C(=O)O)c(N2C(=O)CCC2=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
GRM4 Q14833 1/20 0.39
ALDH1A1 P00352 6/20 0.38
ALOX12 P18054 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
MAPT P10636 2/20 0.37
POLB P06746 2/20 0.37
TP53 P04637 1/20 0.37
KDM4C Q9H3R0 1/20 0.36
MYC P01106 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HPGD P15428 2/20 0.35
ATAD2 Q6PL18 1/20 0.35
CECR2 Q9BXF3 1/20 0.35
STAT3 P40763 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35
CA12 O43570 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7769435 0.87 ALDH1A1 (0.41) KDM4EGRM4ALDH1A1ALOX12MEN1
SCHEMBL27471377 0.85 MYC (0.51) KDM4EGRM4ALDH1A1POLBTP53
SCHEMBL5137956 0.82 ALDH1A1 (0.36) GRM4ALDH1A1ALOX12MEN1KMT2A
SCHEMBL30358600 0.80 ALDH1A1 (0.39) KDM4EALDH1A1ALOX12MEN1KMT2A
Hydrochloric Acid SCHEMBL21800936 0.79 GRM4 (0.39) KDM4EGRM4ALDH1A1MEN1KMT2A
SCHEMBL1232653 0.76 MAPK1 (0.38) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL567033 0.76 KDM4E (0.38) KDM4EGRM4ALDH1A1MEN1KMT2A
SCHEMBL317626 0.74 CA12 (0.42) KDM4EGRM4KMT2ATP53MYC
SCHEMBL26799 0.74 KMT2A (0.58) KDM4EALDH1A1MEN1KMT2AATM
SCHEMBL2898289 0.74 CA12 (0.35) KDM4EALDH1A1KMT2ATP53HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3999 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025151464-A1 ALPHA-PARTICLE RADIONUCLIDE-ANTIBODY CONJUGATES FOR TREATMENT OF SOLID TUMORS THE JOHNS HOPKINS UNIVERSITY (US) 2025-07-17 WO claimed
WO-2025083205-A1 DRUG COMBINATION COMPRISING ANTI-CD37 ANTIBODY MAYTANSINE CONJUGATE AND BCL2 INHIBITOR OR PI3K INHIBITOR DEBIOPHARM INTERNATIONAL S.A. (CH) 2025-04-24 WO claimed
US-20240238432-A1 METHOD FOR GLYCOPROTEIN MODIFICATION HONEYBEAR BIOSCIENCES INC. (TW) 2024-07-18 US claimed
WO-2024151999-A1 POLYMERIZED HEMOGLOBIN SIZE FRACTIONATED VIA TANGENTIAL FLOW FILTRATION OHIO STATE INNOVATION FOUNDATION (US) 2024-07-18 WO claimed
US-20240226312-A1 TREATMENT OF CANCER IN PATIENTS WITH SOLUBLE FR-ALPHA IMMUNOGEN, INC. (US) 2024-07-11 US claimed
WO-2024145600-A1 METHOD FOR GLYCOPROTEIN MODIFICATION HONEYBEAR BIOSCIENCES INC. (TW) 2024-07-04 WO claimed
EP-4347661-A1 TREATMENT OF CANCER IN PATIENTS WITH SOLUBLE FR-ALPHA ImmunoGen, Inc. (US) 2024-04-10 EP claimed
EP-3218410-B1 ANTIBODY DRUG CONJUGATES NOVARTIS AG (CH) 2024-03-27 EP claimed
EP-4313009-A1 MAYTANSINE-ANTIBODY CONJUGATES AND METHODS OF USING SAME Angiex, Inc. (US) 2024-02-07 EP claimed
EP-4309671-A2 METHODS FOR INCREASING EFFICACY OF FOLR1 CANCER THERAPY ImmunoGen, Inc. (US) 2024-01-24 EP claimed
US-5492893-A STERILIZATION OF ANIMALS; THERAPY OD SEX HORMONE RELATEDDISEASES COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1996-02-20 US claimed
US-5488036-A GONADOTROPHINS IN CELLS FOR POLYPEPTIDE HORMONES COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1996-01-30 US claimed
US-5378688-A Conjugating luteinizing hormone releasing hormone to plant, bacterialo or chemical toxins COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 1995-01-03 US claimed
EP-0591369-A1 CAPSID FORMING AND CYSTEIN MODIFIED CHIMAERIC MS2-COAT PROTEIN BTG INTERNATIONAL LIMITED (GB) 1994-04-13 EP claimed
EP-0366770-B1 LIPOSOMES COUPLED TO HORMONES VESTAR INC (US) 1994-02-09 EP claimed
WO-1994000600-A1 SOLID SUPPORTS FOR NUCLEIC ACID HYBRIDIZATION ASSAYS MICROPROBE CORPORATION (US) 1994-01-06 WO claimed
WO-1993000434-A1 CAPSID FORMING AND CYSTEIN MODIFIED CHIMAERIC MS2-COAT PROTEIN BRITISH TECHNOLOGY GROUP LTD. (GB) 1993-01-07 WO claimed
EP-0196669-B1 IMPROVED METHOD OF CONJUGATING METALLOTHIONEIN TO BIOLOGICALLY ACTIVE MOLECULES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-02-12 EP claimed
US-5077210-A Binding of proteins for use as biosensors, bioassays SCIENCE APPLICATIONS INTERNATIONAL CORPORATION 1991-12-31 US claimed
US-4218539-A COUPLING ENZYMES WITH MACROMOLECULES FOR IMMUNOASSAY WELTMAN JOEL K 1980-08-19 US claimed