SCHEMBL4396334

SCHEMBL4396334

COc1cccc2occ(COc3cccc4[nH]c(OC(=O)NC5CCN(CCN6CC[C@H](O)[C@@H](C)C6)CC5)cc34)c12

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.35
ALDH1A1 P00352 5/20 0.35
HSD17B10 Q99714 4/20 0.35
MCHR1 Q99705 4/20 0.33
DRD2 P14416 3/20 0.32
DRD3 P35462 3/20 0.32
HTR2A P28223 2/20 0.32
HPGD P15428 3/20 0.32
MAOB P27338 2/20 0.32
DYRK1A Q13627 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
CCR8 P51685 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
HTR4 Q13639 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4406781 0.93 MAOB (0.34) KDM4EALDH1A1HSD17B10MCHR1DRD2
SCHEMBL2316892 0.93 KDM4E (0.31) KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL4406815 0.92 KDM4E (0.36) KDM4EALDH1A1HSD17B10MCHR1DRD2
SCHEMBL4396521 0.91 DRD2 (0.36) DRD2DRD3HTR2AMAOB
SCHEMBL4398647 0.91 KDM4E (0.33) KDM4EALDH1A1HSD17B10MCHR1HPGD
Hydrochloric Acid SCHEMBL4406708 0.90 HTR1A (0.35) KDM4EALDH1A1HSD17B10MCHR1DRD2
SCHEMBL914445 0.89 KMT2A (0.40) KDM4EALDH1A1HSD17B10DRD2DRD3
SCHEMBL4410352 0.89 KDM4E (0.35) KDM4EALDH1A1DRD2DRD3HTR2A
Hydrochloric Acid SCHEMBL4403444 0.89 HTR7 (0.31) ALDH1A1MCHR1DRD2KMT2A
Hydrochloric Acid SCHEMBL4401793 0.88 FAAH (0.32) ALDH1A1MCHR1MAOBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed