SCHEMBL4396426

SCHEMBL4396426

O=C(NC1CCN(CCN2CCCCCC2)CC1)Oc1cc2c(OCc3coc4ccc(Cl)cc34)cccc2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 2/20 0.37
SOS1 Q07889 5/20 0.37
MAOB P27338 4/20 0.37
MAOA P21397 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTR1A P08908 3/20 0.36
HTR7 P34969 3/20 0.36
HTR2A P28223 3/20 0.35
DRD3 P35462 3/20 0.35
DRD2 P14416 2/20 0.35
CCR5 P51681 1/20 0.35
HTR4 Q13639 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4405864 0.94 SOS1 (0.38) SOS1MAOBMAOAKDM4EALDH1A1
SCHEMBL4396402 0.90 MAOB (0.44) SOS1MAOBMAOAKDM4EALDH1A1
SCHEMBL4410352 0.90 KDM4E (0.35) SOS1MAOBMAOAKDM4EALDH1A1
SCHEMBL4405941 0.89 HTR1A (0.36) BDKRB1SOS1MAOBMAOAHTR1A
SCHEMBL914125 0.88 RHEB (0.42) BDKRB1SOS1MAOBMAOAKDM4E
Hydrochloric Acid SCHEMBL4405568 0.87 ALDH1A1 (0.37) BDKRB1SOS1MAOBMAOAKDM4E
SCHEMBL4403829 0.86 MAOB (0.44) MAOBALDH1A1DRD3DRD2
SCHEMBL4409090 0.86 ALDH1A1 (0.33) SOS1MAOBMAOAKDM4EALDH1A1
Hydrochloric Acid SCHEMBL4405534 0.86 SOS1 (0.38) BDKRB1SOS1MAOBMAOAHTR1A
SCHEMBL4402077 0.85 ALDH1A1 (0.34) SOS1MAOBMAOAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed