SCHEMBL4397630

SCHEMBL4397630

N=C(NO)c1ccc(-n2cccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC2 O75106 2/20 0.50
MAPT P10636 6/20 0.45
RAB9A P51151 4/20 0.45
VHL P40337 1/20 0.44
ELOC Q15369 1/20 0.44
ELOB Q15370 1/20 0.44
LMNA P02545 2/20 0.42
ALDH1A1 P00352 5/20 0.42
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
HPGD P15428 2/20 0.40
CYP1A2 P05177 2/20 0.40
NPC1 O15118 2/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 4/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
MCL1 Q07820 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12348299 0.78 HSD17B10 (0.36) LMNAALDH1A1HPGDCYP2C19
SCHEMBL4399632 0.77 CYP3A4 (0.57) MAPTLMNAMEN1KMT2ATDP1
SCHEMBL3556883 0.75 F2 (0.55) AOC2VHLELOCELOBLMNA
SCHEMBL14174283 0.73 F2 (0.59) MAPTRAB9ALMNAALDH1A1KMT2A
SCHEMBL2361705 0.72 HDAC1 (0.65) RAB9AALDH1A1NPC1SMN1; SMN2L3MBTL1
Benzamidoxime SCHEMBL194059 0.71 HDAC8 (0.50) MAPTALDH1A1MEN1KMT2AHPGD
SCHEMBL8704862 0.69 AOC2 (0.65) AOC2MAPTRAB9ALMNAALDH1A1
SCHEMBL4404636 0.69 HDAC6 (0.61) MAPTRAB9ALMNAALDH1A1MEN1
SCHEMBL771387 0.69 LMNA (0.50) MAPTRAB9ALMNAALDH1A1MEN1
SCHEMBL566487 0.69 CES2 (0.46) RAB9ALMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed