SCHEMBL439833

SCHEMBL439833

COc1ccc(Cl)c2ncc(C(=O)O)c(N)c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.53
CLCN2 P51788 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
DPP4 P27487 1/20 0.38
EGFR P00533 2/20 0.37
KMO O15229 3/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KDM4E B2RXH2 1/20 0.37
FYN P06241 1/20 0.36
SRC P12931 1/20 0.36
TEC P42680 1/20 0.36
BTK Q06187 1/20 0.36
ITK Q08881 1/20 0.36
CSF1R P07333 1/20 0.36
IKBKB O14920 1/20 0.36
PDE5A O76074 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL435825 0.89 HAVCR2 (0.50) HAVCR2CLCN2ALDH1A1MRGPRX4EGFR
SCHEMBL440068 0.84 HAVCR2 (0.63) HAVCR2ALDH1A1KMOKMT2AMAPT
SCHEMBL438246 0.84 DPP4 (0.56) DPP4KMT2AMAPTPDE5AMEN1
SCHEMBL440283 0.81 DYRK1A (0.39) ALDH1A1KMT2AMAPTKDM4EIKBKB
SCHEMBL436999 0.77 NQO2 (0.36) ALDH1A1KMT2AMAPTKDM4EMEN1
SCHEMBL442158 0.76 HAVCR2 (0.54) HAVCR2CLCN2ALDH1A1KMT2AMAPT
SCHEMBL440489 0.74 DPP4 (0.53) DPP4KMT2AMAPTMEN1NPC1
SCHEMBL439862 0.72 HAVCR2 (0.63) HAVCR2KMT2AMEN1
SCHEMBL437260 0.71 HAVCR2 (0.67) HAVCR2ALDH1A1KMT2AMAPTKDM4E
SCHEMBL437796 0.70 NPC1 (0.54) ALDH1A1KMT2AMAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed