SCHEMBL440283

SCHEMBL440283

COc1ccc(Cl)c2ncc(Cl)c(N)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.39
PDPK1 O15530 1/20 0.38
ALDH1A1 P00352 3/20 0.35
HPGD P15428 3/20 0.35
KDM4E B2RXH2 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HIF1A Q16665 1/20 0.35
MAPT P10636 3/20 0.35
NPC1 O15118 2/20 0.35
GAA P10253 2/20 0.35
MAPK1 P28482 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
THRB P10828 1/20 0.35
RAB9A P51151 1/20 0.35
BLM P54132 1/20 0.35
ATM Q13315 1/20 0.35
G6PD P11413 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
KMT2A Q03164 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL439519 0.87 DYRK1A (0.39) DYRK1APDPK1ALDH1A1HPGDKDM4E
SCHEMBL436999 0.86 NQO2 (0.36) DYRK1APDPK1ALDH1A1HPGDKDM4E
SCHEMBL439833 0.81 HAVCR2 (0.53) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL437555 0.80 HAVCR2 (0.38) DYRK1AGAA
SCHEMBL438246 0.76 DPP4 (0.56) MAPTNPC1RAB9AKMT2AMEN1
SCHEMBL438319 0.73 NQO2 (0.36) DYRK1APDPK1ALDH1A1HPGDKDM4E
SCHEMBL441668 0.72 GAA (0.41) DYRK1APDPK1ALDH1A1KDM4EMAPT
SCHEMBL436008 0.72 HTR1A (0.44) ALDH1A1KDM4EG6PD
SCHEMBL437482 0.70 CYP3A4 (0.35) KDM4EMAPTKMT2AMEN1POLB
SCHEMBL435825 0.69 HAVCR2 (0.50) ALDH1A1KDM4EMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed