SCHEMBL4398622

SCHEMBL4398622

C[C@H]1CN([C@@H](C)CN2CCC(NC(=O)Oc3cc4c(OCc5ccoc5)cccc4[nH]3)CC2)CC[C@@H]1O

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.32
MCHR1 Q99705 1/20 0.32
HTR1A P08908 3/20 0.31
SLC6A4 P31645 1/20 0.31
DYRK1A Q13627 1/20 0.31
ACHE P22303 1/20 0.31
PARP1 P09874 1/20 0.31
MEN1 O00255 1/20 0.30
SLC2A1 P11166 1/20 0.30
ADRB3 P13945 2/20 0.30
ADRB2 P07550 1/20 0.30
ADRB1 P08588 1/20 0.30
CCR5 P51681 1/20 0.30
SRD5A2 P31213 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399335 1.00 KMT2A (0.32) KMT2AMCHR1HTR1ASLC6A4DYRK1A
SCHEMBL4411341 0.91 HTR1A (0.34) KMT2AMCHR1HTR1ASLC6A4ACHE
SCHEMBL915392 0.89 KMT2A (0.40) KMT2AHTR1ADYRK1AACHEPARP1
SCHEMBL913688 0.89 KMT2A (0.40) KMT2AHTR1ADYRK1AACHEPARP1
SCHEMBL4405956 0.89 FAAH (0.34) KMT2AMCHR1DYRK1AMEN1CCR5
SCHEMBL4406699 0.89 KMT2A (0.34) KMT2AMCHR1HTR1ASLC6A4ACHE
SCHEMBL4396316 0.89 KMT2A (0.34) KMT2AMCHR1HTR1ASLC6A4ACHE
SCHEMBL4396436 0.86 DRD2 (0.33) HTR1ASLC6A4ACHEADRB3ADRB2
SCHEMBL4410335 0.86 MCHR1 (0.33) KMT2AMCHR1HTR1ASLC6A4DYRK1A
SCHEMBL4405858 0.86 PARP1 (0.34) KMT2AHTR1ASLC6A4DYRK1APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed