SCHEMBL4400748

SCHEMBL4400748

COc1cc(OC)c2c(COc3cccc4[nH]c(OC(=O)NC5CCN(CCN6CCC(O)CC6)CC5)cc34)coc2c1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.37
MCHR1 Q99705 2/20 0.37
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
POLB P06746 2/20 0.34
CD274 Q9NZQ7 1/20 0.34
SIGMAR1 Q99720 7/20 0.33
CCR8 P51685 1/20 0.33
USP2 O75604 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTR4 Q13639 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4406815 0.93 KDM4E (0.36) MAOBMCHR1DRD2DRD3CD274
SCHEMBL4400742 0.92 MCHR1 (0.36) MAOBMCHR1POLBSIGMAR1USP2
Hydrochloric Acid SCHEMBL4406781 0.92 MAOB (0.34) MAOBMCHR1DRD2DRD3POLB
SCHEMBL4401840 0.90 MAOB (0.44) MAOBMCHR1DRD2DRD3SIGMAR1
SCHEMBL4409300 0.89 MAOB (0.44) MAOBMCHR1DRD2DRD3SIGMAR1
SCHEMBL914118 0.89 DRD2 (0.41) MAOBMCHR1DRD2DRD3POLB
Hydrochloric Acid SCHEMBL4406795 0.86 HTR1A (0.39) MCHR1DRD2DRD3CCR8KMT2A
SCHEMBL4405632 0.86 MAOB (0.38) MAOBDRD2DRD3MAOA
SCHEMBL4394210 0.86 MCHR1 (0.34) MAOBMCHR1KMT2AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL4396580 0.86 HTR7 (0.33) MAOBMCHR1DRD2DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed