SCHEMBL4401840

SCHEMBL4401840

COc1ccc2c(COc3cccc4[nH]c(OC(=O)NC5CCN(CCN6CCC(O)CC6)CC5)cc34)coc2c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.44
MCHR1 Q99705 2/20 0.39
LTA4H P09960 3/20 0.38
ALDH1A1 P00352 5/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
SIGMAR1 Q99720 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HTR1A P08908 1/20 0.37
MAPT P10636 2/20 0.37
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4409300 0.94 MAOB (0.44) MAOBMCHR1SIGMAR1DRD2DRD3
SCHEMBL4403829 0.94 MAOB (0.44) MAOBMCHR1LTA4HALDH1A1MEN1
SCHEMBL4399337 0.92 MAOB (0.41) MAOBMCHR1LTA4HALDH1A1SIGMAR1
SCHEMBL4400748 0.90 MAOB (0.37) MAOBMCHR1ALDH1A1KMT2ASIGMAR1
Hydrochloric Acid SCHEMBL4401842 0.90 MCHR1 (0.36) MCHR1SIGMAR1HTR1ADRD2DRD3
SCHEMBL4405941 0.90 HTR1A (0.36) MAOBLTA4HKMT2AHTR1ADRD2
SCHEMBL4405632 0.90 MAOB (0.38) MAOBDRD2DRD3
SCHEMBL4398599 0.89 ALDH1A1 (0.34) MAOBMCHR1LTA4HALDH1A1KMT2A
SCHEMBL4396402 0.89 MAOB (0.44) MAOBMCHR1ALDH1A1MEN1LMNA
SCHEMBL914272 0.89 MAOB (0.47) MAOBMCHR1LTA4HALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed