SCHEMBL440237

SCHEMBL440237

Cc1cc2c(N)cc(-c3ccccc3)nc2cc1Br

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.59
ADORA2A P29274 3/20 0.51
ADORA1 P30542 3/20 0.51
SLC2A1 P11166 1/20 0.50
DHFR P00374 1/20 0.43
CHEK1 O14757 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CCNA1 P78396 1/20 0.43
SMN1; SMN2 Q16637 5/20 0.42
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
PDGFRB P09619 1/20 0.42
KDR P35968 1/20 0.42
FLT3 P36888 1/20 0.42
NCF1 P14598 1/20 0.41
LMNA P02545 2/20 0.41
HPGD P15428 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
KDM4E B2RXH2 6/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL437369 0.78 ACHE (0.67) ACHEADORA2AADORA1SLC2A1SMN1; SMN2
SCHEMBL438920 0.77 ACHE (0.70) ACHEADORA2AADORA1SLC2A1SMN1; SMN2
SCHEMBL27469565 0.77 ACHE (0.70) ACHEADORA2AADORA1SMN1; SMN2RAB9A
SCHEMBL2873300 0.76 ACHE (1.00) ACHEADORA2AADORA1SLC2A1SMN1; SMN2
SCHEMBL4824379 0.74 ACHE (0.71) ACHEADORA2AADORA1SMN1; SMN2RAB9A
SCHEMBL437545 0.73 ADORA1 (0.55) ACHEADORA2AADORA1SLC2A1CHEK1
SCHEMBL437510 0.73 RXFP1 (0.52) ACHEADORA2AADORA1SLC2A1SMN1; SMN2
SCHEMBL439581 0.73 ACHE (0.51) ACHEADORA2AADORA1SLC2A1CHEK1
SCHEMBL28516025 0.73 ACHE (0.93) ACHEADORA2AADORA1SLC2A1SMN1; SMN2
SCHEMBL4143397 0.72 ACHE (0.77) ACHEADORA2AADORA1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed