SCHEMBL437545

SCHEMBL437545

Cc1c(Br)ccc2c(N)cc(-c3ccccc3)nc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.55
ADORA2A P29274 4/20 0.55
EPRS1 P07814 2/20 0.53
ACHE P22303 2/20 0.51
PPARA Q07869 1/20 0.45
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
RAB9A P51151 2/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41
CHEK1 O14757 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CCNA1 P78396 1/20 0.40
NCF1 P14598 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436729 0.80 ACHE (0.60) ADORA1ADORA2AACHEMEN1KMT2A
SCHEMBL439581 0.79 ACHE (0.51) ADORA1ADORA2AACHEMEN1KMT2A
SCHEMBL438193 0.78 NR4A2 (0.51) ADORA1ADORA2AEPRS1MEN1KMT2A
SCHEMBL437510 0.77 RXFP1 (0.52) ADORA1ADORA2AACHEMEN1KMT2A
SCHEMBL440069 0.73 NOS2 (0.41) EPRS1ALDH1A1
SCHEMBL440237 0.73 ACHE (0.59) ADORA1ADORA2AACHEMEN1KMT2A
SCHEMBL438920 0.71 ACHE (0.70) ADORA1ADORA2AEPRS1ACHEMEN1
SCHEMBL27469565 0.71 ACHE (0.70) ADORA1ADORA2AACHEMEN1KMT2A
SCHEMBL22136019 0.71 ACHE (0.51) ADORA1ADORA2AACHEALDH1A1KDM4E
SCHEMBL117482 0.70 EPRS1 (1.00) EPRS1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed