SCHEMBL4403760

SCHEMBL4403760

Cc1nc(COc2cccc3[nH]c(OC(=O)NC4CCN(CC5CCCN6CCCCC56)CC4)cc23)cs1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32
HTR2B P41595 1/20 0.32
ALOX5 P09917 1/20 0.31
LMNA P02545 1/20 0.31
MCHR1 Q99705 1/20 0.31
PARP1 P09874 1/20 0.30
PARP2 Q9UGN5 1/20 0.30
PKM P14618 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963683 0.89 KMT2A (0.37) L3MBTL1ALDH1A1LMNAPARP1PARP2
Hydrochloric Acid SCHEMBL4405691 0.83 LMNA (0.37) ALDH1A1TDP1KDM4ETSHRHTT
SCHEMBL4400753 0.83 ALDH1A1 (0.38) ALDH1A1TDP1KDM4ETSHRHTT
SCHEMBL4411388 0.82 CHRM2 (0.34) ALDH1A1TDP1KDM4ETSHRHTT
SCHEMBL4404600 0.82 ALDH1A1 (0.36) ALDH1A1TDP1KDM4ETSHRHTT
Hydrochloric Acid SCHEMBL4406718 0.81 ALDH1A1 (0.32) ALDH1A1TDP1KDM4ETSHRHTT
Hydrochloric Acid SCHEMBL4397030 0.80 DRD2 (0.35) ALDH1A1TDP1KDM4ETSHRHTT
SCHEMBL4404574 0.80 ALDH1A1 (0.34) ALDH1A1TDP1KDM4ETSHRHTT
Hydrochloric Acid SCHEMBL4406706 0.80 ALDH1A1 (0.34) ALDH1A1TDP1KDM4ETSHRHTT
SCHEMBL4396348 0.79 SOS1 (0.34) ALDH1A1TDP1TSHRHTTSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed