SCHEMBL4411388

SCHEMBL4411388

O=C(NC1CCN(C[C@@H]2CCCN3CCCC[C@H]23)CC1)Oc1cc2c(OCc3ccoc3)cccc2[nH]1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
SRD5A2 P31213 1/20 0.32
LMNA P02545 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
MCHR1 Q99705 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL914948 0.89 KMT2A (0.39) CHRM2CHRM1CHRM3ALDH1A1TDP1
SCHEMBL4403746 0.87 CHRM2 (0.36) CHRM2CHRM1CHRM3KMT2AMEN1
SCHEMBL4400753 0.85 ALDH1A1 (0.38) ALDH1A1TDP1TSHRHTTKDM4E
Hydrochloric Acid SCHEMBL4397030 0.85 DRD2 (0.35) ALDH1A1TDP1TSHRHTTKDM4E
Hydrochloric Acid SCHEMBL4405691 0.84 LMNA (0.37) ALDH1A1TDP1TSHRHTTLMNA
SCHEMBL4396348 0.84 SOS1 (0.34) ALDH1A1TDP1TSHRHTTMAOA
SCHEMBL4409082 0.84 SRD5A2 (0.36) CHRM2CHRM1CHRM3KMT2AMEN1
Hydrochloric Acid SCHEMBL4394242 0.83 TDP1 (0.37) ALDH1A1TDP1TSHRHTTLMNA
Hydrochloric Acid SCHEMBL4406718 0.83 ALDH1A1 (0.32) ALDH1A1TDP1TSHRHTTLMNA
Hydrochloric Acid SCHEMBL4406711 0.83 TDP1 (0.32) ALDH1A1TDP1TSHRHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed