SCHEMBL440378

SCHEMBL440378

Nc1c(C(=O)O)cnc2cc(Cl)cc(Cl)c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 1/20 0.49
AKR1C4 P17516 1/20 0.42
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
AKR1C1 Q04828 1/20 0.42
CYP3A4 P08684 1/20 0.41
POLB P06746 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
TSHR P16473 2/20 0.40
CASP1 P29466 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GABRP O00591 2/20 0.39
GABRD O14764 2/20 0.39
GABRA1 P14867 2/20 0.39
GABRB1 P18505 2/20 0.39
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA5 P31644 2/20 0.39
GABRA3 P34903 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7047957 0.83 AKR1C2 (0.51) HAVCR2AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL29617335 0.83 AKR1C2 (0.51) HAVCR2AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL440854 0.79 AURKA (0.57) SMN1; SMN2KMT2AAURKAAURKBKDM4E
SCHEMBL435967 0.78 NR4A2 (0.38) CYP3A4TSHRAURKAAURKBALDH1A1
SCHEMBL438978 0.75 HAVCR2 (0.64) HAVCR2AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL438230 0.73 NR4A2 (0.35) KMT2AAURKAAURKBHTT
SCHEMBL9389667 0.73 KMO (0.40) SMN1; SMN2KMT2AALDH1A1MEN1MAPT
SCHEMBL7691286 0.72 MAPK1 (0.42) AKR1C4AKR1C3AKR1C2AKR1C1CYP3A4
SCHEMBL442311 0.72 KDM4E (0.40) HAVCR2GABRPGABRDGABRA1GABRB1
SCHEMBL440411 0.72 HAVCR2 (0.52) HAVCR2TSHRCASP1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed