SCHEMBL4406466

SCHEMBL4406466

CC(=O)c1cc(=O)nc2sc(C)nn12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.45
KDM4E B2RXH2 5/20 0.45
HSD17B10 Q99714 5/20 0.43
GAA P10253 1/20 0.43
ALOX15 P16050 1/20 0.43
LMNA P02545 2/20 0.40
TSHR P16473 1/20 0.40
GRIA2 P42262 2/20 0.37
GRIN1 Q05586 2/20 0.37
GRIN2A Q12879 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA3 P07451 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
CA5A P35218 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA13 Q8N1Q1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23415102 0.70 L3MBTL1 (0.65) ALDH1A1KDM4EHSD17B10LMNAGRIA2
SCHEMBL18347279 0.69 RAB9A (0.60) ALDH1A1KDM4EHSD17B10GRIA2GRIN1
SCHEMBL2673777 0.67 NPC1 (0.48) ALDH1A1KDM4EHSD17B10LMNAGRIA2
SCHEMBL11374859 0.65 ALDH1A1 (0.43) ALDH1A1KDM4EHSD17B10GAAALOX15
SCHEMBL2445247 0.65 CA12 (0.39) ALDH1A1KDM4EHSD17B10GAAALOX15
SCHEMBL23415126 0.64 ALPI (0.67)
SCHEMBL12292813 0.63 HSD17B10 (0.47) ALDH1A1KDM4EHSD17B10ALOX15LMNA
SCHEMBL4403129 0.63 CA12 (0.38) ALDH1A1KDM4EHSD17B10GAAALOX15
SCHEMBL11375468 0.62 ALDH1A1 (0.57) ALDH1A1KDM4EHSD17B10GAAALOX15
SCHEMBL3519572 0.62 CA12 (0.57) KDM4EHSD17B10LMNATSHRGRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120107273-A1 NEW PIPERAZINE COMPOUND AND USE THEREOF AS A HCV POLYMERASE INHIBITOR JAPAN TOBACCO INC. (JP) 2012-05-03 US disclosed
US-8017612-B2 therapeutic agent for hepatitis C; R)-4-(4-trifluoromethyl-benzenesulfonyl)-piperazine-1,3-dicarboxylic acid 3-(4-isopropyl-benzylamide) 1-pyridin-4-ylamide; enzyme inhibitors JAPAN TOBACCO INC. (JP) 2011-09-13 US disclosed
US-20080081818-A1 therapeutic agent for hepatitis C; R)-4-(4-trifluoromethyl-benzenesulfonyl)-piperazine-1,3-dicarboxylic acid 3-(4-isopropyl-benzylamide) 1-pyridin-4-ylamide; enzyme inhibitors JAPAN TOBACCO INC. (JP) 2008-04-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080081818-A1 therapeutic agent for hepatitis C; R)-4-(4-trifluoromethyl-benzenesulfonyl)-piperazine-1,3-dicarboxylic acid 3-(4-isopropyl-benzylamide) 1-pyridin-4-ylamide; enzyme inhibitors HAVCR2, AADAC, DNPEP ALDH1A1 96/4885KDM4E 502/4885HSD17B10 1395/4885
US-20120107273-A1 NEW PIPERAZINE COMPOUND AND USE THEREOF AS A HCV POLYMERASE INHIBITOR POLR1C, POLR2E, POLR2H ALDH1A1 557/4885KDM4E 1378/4885HSD17B10 1248/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.