SCHEMBL4409346

SCHEMBL4409346

O=C(NCCNCc1ccc(OCC(F)(F)F)nc1)c1c[nH]c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.46
HTR2C P28335 5/20 0.45
DGAT1 O75907 2/20 0.45
EPHX2 P34913 1/20 0.44
SSTR3 P32745 1/20 0.43
HDAC1 Q13547 3/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
FAAH O00519 1/20 0.42
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4300137 0.87 TRPV1 (0.60) TRPV1HTR2CDGAT1EPHX2HDAC1
SCHEMBL4407981 0.80 DGAT1 (0.47) HTR2CDGAT1EPHX2HDAC1HDAC2
SCHEMBL4406451 0.79 DGAT1 (0.52) DGAT1EPHX2HDAC1HDAC2SCN9A
SCHEMBL4407117 0.77 DGAT1 (0.49) DGAT1EPHX2SCN9A
SCHEMBL4296664 0.75 EPHX2 (0.52) TRPV1HTR2CDGAT1EPHX2HDAC1
SCHEMBL4401623 0.70 DGAT1 (0.57) DGAT1EPHX2HDAC1SCN9A
SCHEMBL4553345 0.70 DGAT1 (0.58) TRPV1DGAT1EPHX2SCN9A
SCHEMBL6204945 0.70 CFTR (0.53) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL7960871 0.69 HDAC1 (0.60) SSTR3HDAC1HDAC2HDAC3HDAC4
SCHEMBL13611460 0.69 DGAT1 (0.62) TRPV1DGAT1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044055-A2 AMIDE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-04-08 EP disclosed
WO-2008011131-A2 AMIDE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-01-24 WO disclosed