SCHEMBL4411564

SCHEMBL4411564

Nc1[nH]c(Nc2ccc3cn[nH]c3c2)nc2ncnc1-2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.49
ALDH1A1 P00352 6/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
HIF1A Q16665 1/20 0.45
PHLPP2 Q6ZVD8 1/20 0.45
HSD17B10 Q99714 1/20 0.45
EIF2AK2 P19525 1/20 0.44
RET P07949 1/20 0.43
KDR P35968 1/20 0.43
MKNK1 Q9BUB5 2/20 0.43
DAPK3 O43293 1/20 0.42
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
PAK4 O96013 1/20 0.42
PIM1 P11309 1/20 0.42
PRKACA P17612 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4428827 0.77 EGFR (0.50) KDRFLT3SYKMAPTRAB9A
SCHEMBL4414311 0.76 EGFR (0.53) ALDH1A1KDRSYKMAPTKMT2A
SCHEMBL4417948 0.75 GAA (0.43) RETKDRDAPK3PRKD3MAP4K4
SCHEMBL4427810 0.74 EGFR (0.45) CYP3A4SYKMAPTKMT2AMEN1
SCHEMBL4414428 0.74 EGFR (0.47) HIF1AHSD17B10HTTRAB9AEGFR
SCHEMBL4413885 0.74 FYN (0.46) ALDH1A1HSD17B10RETKDRDAPK3
SCHEMBL1306611 0.73 IRAK4 (0.45) CDC7RETKDRDAPK3PRKD3
SCHEMBL30250674 0.72 CDC7 (0.70) CDC7ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL4412315 0.71 ABCG2 (0.44) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL4412618 0.71 EGFR (0.49) RETKDRMAP4K4CDK7DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601713-B2 Kinase inhibitors and their uses RIGEL PHARMACEUTICALS, INC. (US) 2009-10-13 US claimed