SCHEMBL4416102

SCHEMBL4416102

[CH2]CNC(=O)c1cc(S(N)(=O)=O)c(Cl)cc1NCc1ccco1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 7/20 0.77
CA1 P00915 7/20 0.77
CA2 P00918 7/20 0.77
CA9 Q16790 7/20 0.77
CA6 P23280 6/20 0.77
CA7 P43166 6/20 0.77
CA14 Q9ULX7 6/20 0.77
CA5B Q9Y2D0 6/20 0.77
CA5A P35218 5/20 0.77
CISD1 Q9NZ45 3/20 0.77
ALDH1A1 P00352 1/20 0.77
HTR1A P08908 1/20 0.77
CA4 P22748 1/20 0.77
HSD11B1 P28845 1/20 0.77
SLC10A1 Q14973 1/20 0.77
GPR35 Q9HC97 1/20 0.77
ABCG2 Q9UNQ0 1/20 0.77
APP P05067 9/20 0.62
CA3 P07451 5/20 0.61
CA13 Q8N1Q1 5/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29436031 0.91 CA12 (0.76) CA12CA1CA2CA9CA6
SCHEMBL10837475 0.90 CA12 (0.82) CA12CA1CA2CA9CA6
SCHEMBL14369223 0.90 CA12 (0.74) CA12CA1CA2CA9CA6
SCHEMBL2880956 0.89 CA12 (0.83) CA12CA1CA2CA9CA6
SCHEMBL29436046 0.89 CA1 (0.79) CA12CA1CA2CA9CA6
SCHEMBL229073 0.88 CA12 (0.85) CA12CA1CA2CA9CA6
Furosemide SCHEMBL428921 0.87 CISD1 (1.00) CA12CA1CA2CA9CA6
Furosemide SCHEMBL29406913 0.87 CISD1 (1.00) CA12CA1CA2CA9CA6
Furosemide SCHEMBL9811 0.87 CISD1 (1.00) CA12CA1CA2CA9CA6
Furosemide SCHEMBL6751172 0.86 CISD1 (0.98) CA12CA1CA2CA9CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1668008-A4 NITROSATED AD NITROSYLATED DIURETIC COMPOUDS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2009-02-25 EP claimed
EP-1668008-A2 NITROSATED AD NITROSYLATED DIURETIC COMPOUDS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2006-06-14 EP claimed
WO-2005023183-A2 NITROSATED AD NITROSYLATED DIURETIC COMPOUDS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2005-03-17 WO claimed
US-20050059655-A1 Nitrosated and nitrosylated diuretic compounds, compositions and methods of use NITROMED, INC. (US) 2005-03-17 US claimed
EP-1668008-A4 NITROSATED AD NITROSYLATED DIURETIC COMPOUDS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2009-02-25 EP disclosed
US-7282519-B2 Nitrosated and nitrosylated diuretic compounds, compositions and methods of use NITROMED, INC. (US) 2007-10-16 US disclosed
EP-1668008-A2 NITROSATED AD NITROSYLATED DIURETIC COMPOUDS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2006-06-14 EP disclosed
WO-2005023183-A2 NITROSATED AD NITROSYLATED DIURETIC COMPOUDS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2005-03-17 WO disclosed
US-20050059655-A1 Nitrosated and nitrosylated diuretic compounds, compositions and methods of use NITROMED, INC. (US) 2005-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050059655-A1 Nitrosated and nitrosylated diuretic compounds, compositions and methods of use REN, NOS1, NOS3 CA12 1897/4885CA1 1129/4885CA2 489/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.