SCHEMBL4420125

SCHEMBL4420125

O=C(O)Cc1ccc(C(=O)CCl)s1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.58
KMT2A Q03164 4/20 0.58
L3MBTL1 Q9Y468 4/20 0.58
TDP1 Q9NUW8 4/20 0.58
POLB P06746 3/20 0.58
RECQL P46063 2/20 0.58
APEX1 P27695 1/20 0.58
HPGD P15428 4/20 0.57
ALDH1A1 P00352 4/20 0.57
NPC1 O15118 1/20 0.57
HTT P42858 1/20 0.57
RAB9A P51151 1/20 0.57
GSK3B P49841 7/20 0.56
BLM P54132 1/20 0.54
MEN1 O00255 2/20 0.53
USP2 O75604 1/20 0.53
HSD17B10 Q99714 1/20 0.53
APOBEC3A P31941 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
ERAP1 Q9NZ08 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9067494 0.80 HPGD (0.65) MAPTKMT2AL3MBTL1TDP1POLB
SCHEMBL4422452 0.80 MAPT (0.59) MAPTKMT2AL3MBTL1TDP1POLB
SCHEMBL3930128 0.79 RAB9A (0.63) MAPTKMT2ATDP1POLBHPGD
SCHEMBL68973 0.77 HPGD (0.59) MAPTKMT2AL3MBTL1TDP1POLB
SCHEMBL1707142 0.77 HPGD (0.61) MAPTKMT2AL3MBTL1TDP1POLB
SCHEMBL11626640 0.76 HPGD (0.50) MAPTKMT2AL3MBTL1TDP1POLB
Methane SCHEMBL7759142 0.76 HPGD (0.59) MAPTKMT2AL3MBTL1TDP1POLB
SCHEMBL11680962 0.76 KMT2A (0.59) MAPTKMT2AL3MBTL1TDP1POLB
SCHEMBL10520514 0.75 ALDH1A1 (0.54) MAPTL3MBTL1TDP1POLBRECQL
SCHEMBL14190598 0.74 MAPT (0.50) MAPTKMT2AL3MBTL1TDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682538-A4 BIARYL LINKED HYDROXAMATES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S BIO PTE LTD (SG) 2009-05-27 EP disclosed
US-20070167499-A1 Biaryl linked hydroxamates: preparation and pharmaceutical applications A*BIO PTE LTD. (SG) 2007-07-19 US disclosed
US-20070167499-A1 Biaryl linked hydroxamates: preparation and pharmaceutical applications A*BIO PTE LTD. (SG) 2007-07-19 US disclosed
US-20070167499-A1 Biaryl linked hydroxamates: preparation and pharmaceutical applications A*BIO PTE LTD. (SG) 2007-07-19 US disclosed
EP-1682538-A1 BIARYL LINKED HYDROXAMATES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S*Bio Pte Ltd (SG) 2006-07-26 EP disclosed
WO-2005040161-A1 BIARYL LINKED HYDROXAMATES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S*BIO PTE LTD (SG) 2005-05-06 WO disclosed
WO-2005040161-A1 BIARYL LINKED HYDROXAMATES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S*BIO PTE LTD (SG) 2005-05-06 WO disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed
WO-1996004282-A1 CARBAPENEM COMPOUNDS, COMPOSITIONS AND METHODS OF TREATMENT MERCK & CO., INC. (US) 1996-02-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167499-A1 Biaryl linked hydroxamates: preparation and pharmaceutical applications HDAC1, HDAC11, HDAC2 MAPT 3965/4885KMT2A 80/4885L3MBTL1 2252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.