SCHEMBL4421143

SCHEMBL4421143

C1=CN=C(N2CCNCC2)NC=C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.40
PLD1 Q13393 2/20 0.40
NCF1 P14598 1/20 0.40
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 1/20 0.36
ADRB1 P08588 4/20 0.34
HTR3E A5X5Y0 3/20 0.34
HTR3B O95264 3/20 0.34
HTR3A P46098 3/20 0.34
HTR3D Q70Z44 3/20 0.34
HTR3C Q8WXA8 3/20 0.34
SIGMAR1 Q99720 2/20 0.34
LMNA P02545 1/20 0.34
HRH1 P35367 1/20 0.34
CASP1 P29466 1/20 0.33
CASP4 P49662 1/20 0.33
CASP5 P51878 1/20 0.33
USP2 O75604 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL726036 0.83 ADRB2 (0.41) ADRB2PLD1NCF1ALDH1A1KDM4E
SCHEMBL3712448 0.80 CHRNB2 (0.33) CHRNB2CHRNA4
SCHEMBL13611642 0.68 ADRB2 (0.46) ADRB2PLD1NCF1ALDH1A1KDM4E
SCHEMBL2066449 0.67 ADRB1 (0.38) ADRB2PLD1NCF1ALDH1A1KDM4E
SCHEMBL4418589 0.66 ADRB2 (0.35) ADRB2PLD1NCF1ALDH1A1KDM4E
SCHEMBL1420015 0.65 ADRB1 (0.36) ADRB2PLD1NCF1ALDH1A1KDM4E
SCHEMBL726035 0.64 ADRB2 (0.37) ADRB2PLD1NCF1ALDH1A1KDM4E
SCHEMBL27511861 0.62 ADRB2 (0.36) ADRB2PLD1NCF1ALDH1A1KDM4E
SCHEMBL3833595 0.62 ADRB1 (0.39) NCF1ALDH1A1KDM4EADRB1HTR3E
SCHEMBL2175146 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1696931-B1 AMINO SUBSTITUTED DIARYL[A,D]CYCLOHEPTENE ANALOGS AS MUSCARINIC AGONISTS AND METHODS OF TREATMENT OF NEUROPSYCHIATRIC DISORDERS ACADIA PHARM INC (US) 2009-03-25 EP disclosed