SCHEMBL3712448

SCHEMBL3712448

C1=CN=C(N2CCCNC2)NC=C1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 9/20 0.33
CHRNA4 P43681 9/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4421143 0.80 ADRB2 (0.40) CHRNB2CHRNA4
SCHEMBL2304918 0.70
SCHEMBL1533833 0.70 CHRNB2 (0.30) CHRNB2CHRNA4
SCHEMBL15676839 0.65 CHRNB2 (0.46) CHRNB2CHRNA4
SCHEMBL726036 0.63 ADRB2 (0.41) CHRNB2CHRNA4
SCHEMBL6631277 0.60 CHRNB2 (0.37) CHRNB2CHRNA4
SCHEMBL2051022 0.59 HTR3A (0.57) CHRNB2CHRNA4
SCHEMBL9881497 0.58 CHRNB2 (0.54) CHRNB2CHRNA4
SCHEMBL20255363 0.58 CHRNB2 (0.54) CHRNB2CHRNA4
SCHEMBL22538719 0.58 HTR1A (0.41) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110214142-B Tetracyclic heterocyclic compounds useful as HIV integrase inhibitors 默沙东公司 2022-04-01 CN disclosed
EP-2391212-A1 BRIDGED COMPOUNDS AS HIV INTEGRASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2011-12-07 EP disclosed
WO-2010088167-A1 BRIDGED COMPOUNDS AS HIV INTEGRASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-08-05 WO disclosed