SCHEMBL4424979

SCHEMBL4424979

CNC(=O)Cn1c(=O)oc2cc(Br)c(Cl)cc21

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMO O15229 6/20 0.47
KMT2A Q03164 5/20 0.45
MEN1 O00255 4/20 0.45
POLB P06746 3/20 0.45
TP53 P04637 2/20 0.45
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
HSD17B10 Q99714 1/20 0.42
IDO1 P14902 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4425116 0.79 KMT2A (0.66) KMOKMT2AMEN1POLBTP53
SCHEMBL4414447 0.79 TP53 (0.67) KMT2AMEN1POLBTP53ALDH1A1
SCHEMBL4411764 0.79 TP53 (0.61) KMT2AMEN1POLBTP53ALDH1A1
SCHEMBL16836587 0.78 KMO (0.59) KMO
SCHEMBL16836516 0.76 KMO (0.80) KMO
SCHEMBL4427310 0.72 LMNA (0.71) KMT2AMEN1POLBTP53LMNA
SCHEMBL9715993 0.71 KMO (0.43) KMOKMT2AIDO1
Tromethamine SCHEMBL16836500 0.69 KMO (0.77) KMO
SCHEMBL16836502 0.66 KMO (0.57) KMO
SCHEMBL4414327 0.66 KMT2A (0.62) KMOKMT2AMEN1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293775-B2 Benzoxazolone derivatives, processes for preparing them and their uses UCB PHARMA, S.A. (BE) 2012-10-23 US disclosed
EP-1756071-B1 BENZOXAZOLONE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA SA (BE) 2009-08-26 EP disclosed
US-20070299118-A1 Benzoxazolone Derivatives, Processes For Preparing Them And Their Uses UCB, S.A. (BE) 2007-12-27 US disclosed
EP-1756071-A1 BENZOXAZOLONE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB, S.A. (BE) 2007-02-28 EP disclosed
WO-2005118561-A1 BENZOXAZOLONE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB, S.A. (BE) 2005-12-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070299118-A1 Benzoxazolone Derivatives, Processes For Preparing Them And Their Uses PARK7, SNCA, GABRA5 KMO 67/4885KMT2A 2566/4885MEN1 4642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.