SCHEMBL442622

SCHEMBL442622

Cc1cc(C)cc(-c2cc3c(-c4ccccc4)n(-c4ccccc4)c(-c4ccccc4)c3cc2-c2cc(C)cc(C)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD9 Q9H8M2 1/20 0.41
BRD7 Q9NPI1 1/20 0.41
MAPK1 P28482 2/20 0.37
RECQL P46063 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
POLB P06746 1/20 0.37
AVPR1A P37288 1/20 0.37
TSHR P16473 2/20 0.36
PSMB5 P28074 1/20 0.36
KMT2A Q03164 5/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2D6 P10635 1/20 0.36
SSTR2 P30874 1/20 0.36
IL1R1 P14778 1/20 0.36
MEN1 O00255 4/20 0.35
KDM4E B2RXH2 2/20 0.35
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL444839 0.86 IL1R1 (0.41) MAPK1RECQLSMN1; SMN2POLBAVPR1A
SCHEMBL443170 0.73 KDM4E (0.52) MAPK1RECQLSMN1; SMN2POLBAVPR1A
SCHEMBL445355 0.73 ALDH1A1 (0.48) MAPK1SMN1; SMN2NPC1RAB9ACYP2C9
SCHEMBL444851 0.73 IL1R1 (0.44) MAPK1RECQLSMN1; SMN2POLBAVPR1A
SCHEMBL443111 0.72 GAA (0.51) MAPK1SMN1; SMN2POLBTSHRKMT2A
SCHEMBL17911732 0.72 KMT2A (0.51) MAPK1RECQLSMN1; SMN2POLBAVPR1A
SCHEMBL442621 0.70 ALDH1A1 (0.40) BRD9BRD7RAB9ACYP2C9CYP2C19
SCHEMBL27414909 0.69 CA12 (0.46) BRD9BRD7MAPK1SMN1; SMN2PSMB5
SCHEMBL14595487 0.69 AVPR1A (0.55) MAPK1SMN1; SMN2AVPR1ATSHRKMT2A
SCHEMBL13086978 0.69 L3MBTL1 (0.49) BRD9BRD7MAPK1POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8809543-B2 Electrophotographic photoreceptor, electrophotographic image forming method, electrophotographic image forming apparatus, and process cartridge for electrophotographic image forming apparatus RICOH COMPANY, LTD. (JP) 2014-08-19 US disclosed
US-8809543-B2 Electrophotographic photoreceptor, electrophotographic image forming method, electrophotographic image forming apparatus, and process cartridge for electrophotographic image forming apparatus RICOH COMPANY, LTD. (JP) 2014-08-19 US disclosed
US-20120064443-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, ELECTROPHOTOGRAPHIC IMAGE FORMING METHOD, ELECTROPHOTOGRAPHIC IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE FOR ELECTROPHOTOGRAPHIC IMAGE FORMING APPARATUS RICOH COMPANY, LTD. (JP) 2012-03-15 US disclosed
US-20120064443-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR, ELECTROPHOTOGRAPHIC IMAGE FORMING METHOD, ELECTROPHOTOGRAPHIC IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE FOR ELECTROPHOTOGRAPHIC IMAGE FORMING APPARATUS RICOH COMPANY, LTD. (JP) 2012-03-15 US disclosed