SCHEMBL4427520

SCHEMBL4427520

O=[N+]([O-])c1c[c]c(Br)c(-c2cccc(CC(F)(F)F)c2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
AKR1C3 P42330 3/20 0.33
AKR1C2 P52895 3/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
LMNA P02545 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PAX8 Q06710 1/20 0.32
ALOX5 P09917 1/20 0.32
ORAI1 Q96D31 1/20 0.31
ALDH1A1 P00352 4/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
POLB P06746 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4427523 0.80 PTGES (0.35) ALDH1A1CYP19A1
SCHEMBL4431948 0.74 MEN1 (0.33) MEN1KMT2AORAI1RXFP1KDM4E
SCHEMBL27323340 0.74 TSHR (0.61) TSHRMEN1KMT2ALMNAALDH1A1
SCHEMBL30781045 0.74 TSHR (0.61) TSHRMEN1KMT2ALMNAALDH1A1
SCHEMBL5086477 0.73 ALDH1A1 (0.51) TSHRAKR1C3AKR1C2LMNANPC1
SCHEMBL5085402 0.69 ALDH1A1 (0.39) TSHRMEN1KMT2ALMNAALOX5
SCHEMBL4607416 0.67
SCHEMBL4607420 0.65 EGLN1 (0.30)
SCHEMBL29044683 0.65 ALDH1A1 (0.43) MEN1KMT2AALDH1A1MAPTPOLB
SCHEMBL9474702 0.64 LOXL2 (0.55) TSHRAKR1C3ALDH1A1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121660-A2 FUNGICIDAL AMIDES E. I. Du Pont de Nemours and Company (US) 2009-11-25 EP disclosed
WO-2008091580-A2 FUNGICIDAL AMIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-31 WO disclosed
EP-1948649-A2 FUNGICIDAL CARBOXAMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-30 EP disclosed
WO-2007014290-A2 FUNGICIDAL CARBOXAMIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2007-02-01 WO disclosed