SCHEMBL4433374

SCHEMBL4433374

Cc1nc(Cc2ccc(Cl)cc2)sc1NC(=O)c1ccc2c(c1)CCN(C(=O)O)C2CC(C)C

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 1/20 0.36
PPARA Q07869 6/20 0.35
XDH P47989 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
IDO1 P14902 2/20 0.35
KCNH2 Q12809 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
PTGER1 P34995 1/20 0.35
GAA P10253 1/20 0.34
DGAT1 O75907 1/20 0.34
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433371 0.87 PPARA (0.37) GPR52PPARAXDHSMN1; SMN2KDM4E
SCHEMBL4422309 0.83 GAA (0.52) SMN1; SMN2KDM4EALDH1A1LMNAMAPT
SCHEMBL4277759 0.75 PTGER1 (0.48) GPR52XDHSMN1; SMN2KDM4EALDH1A1
SCHEMBL3856745 0.75 PTGER1 (0.49) SMN1; SMN2MAPTHTTPTGER1
Hydrochloric Acid SCHEMBL4279956 0.75 PTGER1 (0.48) GPR52XDHSMN1; SMN2KDM4EALDH1A1
SCHEMBL4425380 0.74 MTNR1B (0.37) GPR52
SCHEMBL13573316 0.73 ESR2 (0.48) SMN1; SMN2HTTPTGER1
SCHEMBL4022473 0.73 PTGDR2 (0.38) SMN1; SMN2ALDH1A1LMNAMAPTHTT
SCHEMBL3666731 0.72 KDM1A (0.41)
SCHEMBL4553186 0.72 FFAR1 (0.44) SMN1; SMN2LMNAMAPTHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed