SCHEMBL4553186

SCHEMBL4553186

CC(C)CC1c2ccc(NC(=O)c3nnc(Cc4ccc(Cl)c(Cl)c4)s3)cc2CCN1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 12/20 0.44
NOD1 Q9Y239 1/20 0.37
OPRD1 P41143 4/20 0.36
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
WNT3A P56704 1/20 0.34
USP7 Q93009 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4555438 0.87 MTNR1B (0.38) FFAR1
SCHEMBL4553185 0.86 FFAR1 (0.45) FFAR1NOD1MEN1LMNAMAPT
SCHEMBL4554892 0.83 FFAR1 (0.43) FFAR1
SCHEMBL3664741 0.74 SMN1; SMN2 (0.53) NOD1MEN1LMNAMAPTHTT
SCHEMBL3727106 0.74 FFAR1 (0.47) FFAR1MEN1LMNAMAPTHTT
SCHEMBL4555618 0.74 MTNR1B (0.42) MEN1LMNAMAPTHTTRAB9A
Hydrochloric Acid SCHEMBL3725782 0.73 FFAR1 (0.47) FFAR1MEN1LMNAMAPTHTT
SCHEMBL3665398 0.73 ROCK2 (0.44) LMNA
SCHEMBL4555437 0.72 FFAR1 (0.38) FFAR1USP7
SCHEMBL3728485 0.72 ESR2 (0.47) FFAR1NOD1MEN1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125799-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE Smithkline Beecham Corporation (US) 2009-12-02 EP disclosed
WO-2008104524-A1 THIADIAZOLE DERIVATIVES, INHIBITORS OF STEAROYL-COA DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2008-09-04 WO disclosed