SCHEMBL3856745

SCHEMBL3856745

Cc1cc(NC(=O)c2ccc3c(c2)CCN(C(=O)O)C3CC(C)C)nn1Cc1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 17/20 0.49
TP53 P04637 1/20 0.43
P2RY14 Q15391 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3856743 0.86 PTGER1 (0.46) PTGER1TP53P2RY14MAPTHTT
SCHEMBL4795246 0.85 PTGER1 (0.71) PTGER1
SCHEMBL3854465 0.84 PTGER1 (0.46) PTGER1
SCHEMBL3847525 0.84 PTGER1 (0.48) PTGER1
SCHEMBL3844837 0.77 PTGER1 (0.61) PTGER1
SCHEMBL4022473 0.77 PTGDR2 (0.38) TP53MAPTHTTSMN1; SMN2NPSR1
SCHEMBL3177484 0.77 PTGER1 (0.66) PTGER1TP53P2RY14MAPTHTT
SCHEMBL4433374 0.75 GPR52 (0.36) PTGER1MAPTHTTSMN1; SMN2
SCHEMBL4795243 0.74 PTGER1 (0.70) PTGER1
SCHEMBL3186899 0.74 PTGER1 (0.52) PTGER1TP53P2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2106398-A2 ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF STEAROYL-COA DESATURASE (SCD) SmithKline Beecham Corporation (US) 2009-10-07 EP disclosed
WO-2008074832-A2 ISOQUINOLINECARBOXAMIDES AS INHIBITORS OF STEAROYL-COA DESATURASE ( SCD) SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed