SCHEMBL4437878

SCHEMBL4437878

COC(=O)c1ncccc1B(O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.58
ALOX15 P16050 2/20 0.44
MAP2K1 Q02750 1/20 0.44
HTT P42858 1/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 7/20 0.43
TDP1 Q9NUW8 1/20 0.43
NPSR1 Q6W5P4 2/20 0.42
BRD4 O60885 1/20 0.41
PARP1 P09874 1/20 0.40
PKM P14618 1/20 0.39
KDM6B O15054 1/20 0.39
KDM5C P41229 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM2A Q9Y2K7 1/20 0.39
KDM3A Q9Y4C1 1/20 0.39
STAT3 P40763 1/20 0.39
HIF1A Q16665 1/20 0.39
MAPT P10636 2/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29953673 0.81 POLB (0.40) L3MBTL1ALOX15ALDH1A1KDM4ENPSR1
SCHEMBL18705823 0.80 L3MBTL1 (0.46) L3MBTL1ALOX15MAP2K1HTTALDH1A1
SCHEMBL69177 0.79 L3MBTL1 (0.64) L3MBTL1ALOX15MAP2K1HTTALDH1A1
SCHEMBL29416324 0.78 L3MBTL1 (0.62) L3MBTL1ALOX15MAP2K1HTTALDH1A1
SCHEMBL69990 0.78 L3MBTL1 (0.62) L3MBTL1ALOX15MAP2K1HTTALDH1A1
SCHEMBL108876 0.78 L3MBTL1 (0.62) L3MBTL1ALOX15MAP2K1HTTALDH1A1
SCHEMBL128711 0.78 L3MBTL1 (0.62) L3MBTL1ALOX15MAP2K1HTTALDH1A1
SCHEMBL31347575 0.78 L3MBTL1 (0.62) L3MBTL1ALOX15MAP2K1HTTALDH1A1
SCHEMBL2561503 0.77 L3MBTL1 (0.57) L3MBTL1ALOX15MAP2K1HTTALDH1A1
SCHEMBL3461964 0.77 L3MBTL1 (0.52) L3MBTL1ALDH1A1KDM4ETDP1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117534613-A Preparation method of 3-aminopyridine-2-carboxylic acid methyl ester 武威广达科技有限公司 2024-02-09 CN disclosed
EP-2124913-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS Novartis AG (CH) 2009-12-02 EP disclosed
WO-2008077597-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS NOVARTIS AG (CH) 2008-07-03 WO disclosed