SCHEMBL4439829

SCHEMBL4439829

O=C1N[C@@H](c2cccc(C(F)(F)F)c2)CN1c1ccc(Oc2ccc(Cl)cc2)nc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LIPE Q05469 7/20 0.38
MAPT P10636 3/20 0.38
HTT P42858 3/20 0.38
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NPBWR1 P48145 1/20 0.36
MCHR1 Q99705 1/20 0.36
SCN9A Q15858 2/20 0.36
MGLL Q99685 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4439090 0.89 SCN9A (0.42) ALDH1A1MAPTHTTLMNACYP3A4
SCHEMBL4439837 0.89 SCN9A (0.42) ALDH1A1MAPTHTTLMNACYP3A4
SCHEMBL4437663 0.89 SCN9A (0.42) ALDH1A1MAPTHTTLMNACYP3A4
SCHEMBL4439959 0.88 SCN9A (0.38) ALDH1A1POLBL3MBTL1LIPEMAPT
SCHEMBL4439973 0.84 PBRM1 (0.44) ALDH1A1MAPTHTTLMNACYP3A4
SCHEMBL3580835 0.80 ALDH1A1 (0.39) ALDH1A1POLBL3MBTL1LIPEMAPT
SCHEMBL3580839 0.80 ALDH1A1 (0.39) ALDH1A1POLBL3MBTL1LIPEMAPT
SCHEMBL4445493 0.79 LIPE (0.39) ALDH1A1POLBL3MBTL1LIPEMAPT
SCHEMBL4439891 0.78 FNTA (0.38) ALDH1A1MAPTHTTLMNACYP2C9
SCHEMBL4745885 0.78 KMT2A (0.47) ALDH1A1MAPTHTTCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121598-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2009-11-25 EP disclosed
WO-2008076754-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-06-26 WO disclosed