SCHEMBL4440419

SCHEMBL4440419

COc1ccc(C(CC=O)c2ccc(F)cc2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PDE4A P27815 1/20 0.45
ACHE P22303 2/20 0.41
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
MMP1 P03956 1/20 0.40
ALDH1A1 P00352 3/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 1/20 0.40
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
IKBKG Q9Y6K9 1/20 0.39
KDM4E B2RXH2 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441719 0.85 AKR1C3 (0.46) MEN1KMT2AACHEPPARGPPARD
SCHEMBL65457 0.80 CACNA2D1 (0.37) NPSR1
SCHEMBL7873221 0.76 ACHE (0.50) MAPTKMT2ANPSR1ACHEPPARG
SCHEMBL22209150 0.75 BCHE (0.55) MEN1MAPTKMT2ANPSR1ACHE
SCHEMBL8324410 0.75 ACHE (0.49) KMT2ANPSR1PDE4AACHEPPARG
SCHEMBL8334710 0.75 ACHE (0.49) KMT2ANPSR1PDE4AACHEPPARG
SCHEMBL4441784 0.75 ACHE (0.51) MEN1MAPTKMT2ANPSR1PDE4A
SCHEMBL7911236 0.74 PDE4A (0.71) PDE4A
SCHEMBL15577528 0.74 HTR2A (0.41) MEN1MAPTKMT2ANPSR1ALDH1A1
SCHEMBL8323966 0.73 GAA (0.45) NFE2L2KMT2ANPSR1ACHEPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed