SCHEMBL4440973

SCHEMBL4440973

CCOC(=O)ON1CCc2sc(C=O)cc2C1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
GAA P10253 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 4/20 0.32
LMNA P02545 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
KCNQ2 O43526 3/20 0.31
MAPT P10636 2/20 0.31
MAPK1 P28482 1/20 0.31
SLC5A1 P13866 1/20 0.30
SLC5A2 P31639 1/20 0.30
KCNQ3 O43525 1/20 0.30
TDP1 Q9NUW8 2/20 0.30
L3MBTL1 Q9Y468 2/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2921885 0.81 MAPT (0.44) ALDH1A1GAANPSR1MEN1KMT2A
SCHEMBL16038585 0.77 GRM5 (0.43) ALDH1A1GAAKDM4ELMNAMAPT
SCHEMBL7782039 0.72 ALDH1A1 (0.40) ALDH1A1GAANPSR1MEN1KMT2A
SCHEMBL3555661 0.71 NOTUM (0.47) ALDH1A1MEN1KMT2AHDAC6MAPT
SCHEMBL4440822 0.70 PRMT5 (0.38) ALDH1A1GAANPSR1MEN1KMT2A
SCHEMBL2925102 0.70 MAOA (0.40) ALDH1A1KDM4EHDAC6MAPTTDP1
SCHEMBL3441635 0.69 HDAC6 (0.43) ALDH1A1MEN1KMT2AHDAC6MAPT
SCHEMBL2923721 0.68 ESR2 (0.53) KDM4ELMNAHDAC6MAPTMAPK1
SCHEMBL6987113 0.67 PDK1 (0.49) ALDH1A1GAAMEN1KMT2AKDM4E
SCHEMBL2925057 0.66 DRD2 (0.47) ALDH1A1KDM4EMAPK1L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132193-B1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INT (DE) 2012-10-24 EP disclosed
EP-2132193-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS Boehringer Ingelheim International GmbH (DE) 2009-12-16 EP disclosed
WO-2008116881-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-02 WO disclosed