SCHEMBL4444660

SCHEMBL4444660

COc1ccc(COCc2cncc(CC=O)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
IDO1 P14902 2/20 0.41
AGXT P21549 2/20 0.41
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 4/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
ALOX12 P18054 1/20 0.40
EGLN1 Q9GZT9 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3593017 0.79 CYP11B1 (0.43) TDP1NPC1RAB9ACYP11B1CYP11B2
SCHEMBL3967034 0.77 CYP11B1 (0.43) CYP11B1CYP11B2CYP3A4
SCHEMBL17981899 0.77 NPC1 (0.44) HDAC4HDAC6TDP1NPC1RAB9A
SCHEMBL3599665 0.77 CYP1A2 (0.51) HDAC4HDAC6NPC1RAB9ACYP11B1
Formic Acid SCHEMBL6366129 0.76 IDO1 (0.53) HDAC4HDAC6TDP1NPC1RAB9A
SCHEMBL190915 0.75 ALDH1A1 (0.65) IDO1AGXTHTTSMN1; SMN2ALDH1A1
SCHEMBL34413 0.75 IDO1 (0.67) TDP1IDO1AGXTHTTSMN1; SMN2
SCHEMBL3961229 0.74 IDO1 (0.52) TDP1NPC1RAB9AIDO1AGXT
Potassium SCHEMBL1477050 0.73 IDO1 (0.64) TDP1IDO1AGXTHTTSMN1; SMN2
Methoxymethane SCHEMBL28823290 0.73 IDO1 (0.64) TDP1IDO1AGXTHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125778-A1 CERTAIN PYRAZOLINE DERIVATIVES WITH KINASE INHIBITORY ACTIVITY Millennium Pharmaceuticals, Inc. (US) 2009-12-02 EP disclosed
WO-2008079277-A1 CERTAIN PYRAZOLINE DERIVATIVES WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed