SCHEMBL4445019

SCHEMBL4445019

COc1ccccc1N1CCN(CCCCOc2ccc3nccn3c2)CC1.Clc1cccc(N2CCN(CCCCOc3ccc4nccn4c3)CC2)c1Cl

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 17/20 0.60
DRD2 P14416 15/20 0.60
DRD4 P21917 5/20 0.59
DRD1 P21728 2/20 0.59
HTR2A P28223 2/20 0.59
LMNA P02545 2/20 0.55
ALDH1A1 P00352 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
MAPT P10636 1/20 0.55
NLRP1 Q9C000 1/20 0.55
SLC6A2 P23975 1/20 0.55
SLC6A4 P31645 1/20 0.55
ADRA1A P35348 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3617541 0.92 DRD3 (0.68) DRD3DRD2DRD4DRD1HTR2A
SCHEMBL3618645 0.92 DRD2 (0.68) DRD3DRD2DRD4DRD1HTR2A
SCHEMBL3616133 0.87 DRD3 (0.58) DRD3DRD2DRD4DRD1HTR2A
SCHEMBL14494809 0.78 DRD2 (0.66) DRD3DRD2DRD4DRD1HTR2A
SCHEMBL4564124 0.78 DRD2 (0.60) DRD3DRD2DRD4DRD1HTR2A
SCHEMBL4450992 0.78 ALDH1A1 (0.57) DRD3DRD2DRD4DRD1HTR2A
SCHEMBL3615992 0.76 DRD2 (0.69) DRD3DRD2DRD4HTR2A
SCHEMBL14494822 0.76 DRD2 (0.62) DRD3DRD2DRD4HTR2A
SCHEMBL4441972 0.75 DRD2 (0.83) DRD3DRD2DRD4DRD1HTR2A
SCHEMBL1114388 0.75 LMNA (0.64) DRD3DRD2DRD4DRD1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137185-A2 INDOLIZINES AND AZA-ANALOG DERIVATIVES THEREOF AS CNS ACTIVE COMPOUNDS Gmeiner, Dr. Peter (DE) 2009-12-30 EP disclosed
WO-2008113559-A2 INDOLIZINES AND AZA-ANALOG DERIVATIVES THEREOF AS CNS ACTIVE COMPOUNDS SCHWARZ PHARMA AG (DE) 2008-09-25 WO disclosed