SCHEMBL4450951

SCHEMBL4450951

Clc1cccc2c1OC1(CC2)CCN(c2ccc(-c3cccnc3)nn2)CC1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCD O00767 16/20 0.53
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
CNR2 P34972 1/20 0.42
TRPM8 Q7Z2W7 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4445219 0.79 TRPM8 (0.44) SCDCNR2TRPM8
SCHEMBL4556505 0.78 TRPM8 (0.43) SCDCYP3A4CYP2D6TRPM8
SCHEMBL4555897 0.71 CNR2 (0.42) SCDCNR2TRPM8
SCHEMBL4557042 0.71 CNR2 (0.39) CYP2C9CNR2TRPM8
SCHEMBL4136835 0.68 SCD (0.46) SCDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL31629219 0.67 SCD (1.00) SCDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL13930227 0.66 TRPM8 (0.39) SCDCYP3A4CNR2TRPM8
SCHEMBL4566242 0.66 CYP3A4 (0.42) SCDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL13770570 0.65 TRPM8 (0.49) CYP2D6TRPM8
SCHEMBL1742505 0.65 CYP2C9 (0.52) SCDCYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037542-A2 SPIROCYCLIC COMPOUNDS AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-03-26 WO disclosed
WO-2009037542-A2 SPIROCYCLIC COMPOUNDS AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-03-26 WO disclosed