SCHEMBL4454235

SCHEMBL4454235

Nc1cnccc1NCc1nccs1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM5 Q9NZQ8 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDM1A O60341 1/20 0.39
MAOB P27338 1/20 0.39
TLR7 Q9NYK1 1/20 0.37
KDM4C Q9H3R0 2/20 0.36
KDM4E B2RXH2 1/20 0.36
KDM6B O15054 1/20 0.36
KDM4A O75164 1/20 0.36
KDM5C P41229 1/20 0.36
KDM4D Q6B0I6 1/20 0.36
SLCO1B1 Q9Y6L6 1/20 0.36
ROCK2 O75116 1/20 0.35
AOC1 P19801 2/20 0.35
AOC3 Q16853 2/20 0.35
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE1C Q14123 1/20 0.34
NR1H3 Q13133 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30504120 0.74 MAPK10 (0.45) TRPM5KDM4CKDM4EKDM6BKDM4A
SCHEMBL16657366 0.73 ALDH1A1 (0.45) KDM4EALDH1A1TSHRNOS1HSD17B10
SCHEMBL6297758 0.71 CYP2C19 (0.57) TRPM5CYP2C19KDM1AMAOBTLR7
SCHEMBL16489564 0.71 KDM4C (0.56) KDM4CKDM4EKDM6BKDM4AKDM4D
SCHEMBL15722502 0.71 MAOA (0.54) CYP2C19MAOBKDM4EALDH1A1HSD17B10
SCHEMBL22346318 0.71 TRPM5 (0.41) TRPM5CYP2C19KDM1AMAOBTLR7
SCHEMBL20874597 0.71 TRPM5 (0.41) TRPM5CYP2C19KDM1AMAOBTLR7
Hydrochloric Acid SCHEMBL6297635 0.70 CYP2C19 (0.56) TRPM5CYP2C19KDM1AMAOBTLR7
SCHEMBL30703857 0.70 AOC1 (0.56) KDM4EAOC1AOC3ALDH1A1
SCHEMBL9329604 0.70 AOC1 (0.56) KDM4EAOC1AOC3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819000-B1 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2009-07-08 EP disclosed