SCHEMBL44556

SCHEMBL44556

COCCOc1cc(-c2cn3ncccc3n2)cc(-c2noc(C(=O)NCCN3CCCCC3)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 16/20 0.43
PIM1 P11309 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
TSHR P16473 1/20 0.39
SCN9A Q15858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44956 0.93 HSD17B10 (0.43) GSK3B
SCHEMBL43952 0.85 SMPD1 (0.36) GSK3B
SCHEMBL44541 0.85 PDE4B (0.41) TSHR
SCHEMBL44296 0.84 MARK3 (0.39) HDAC4HDAC6
SCHEMBL44205 0.83 SMPD1 (0.35)
SCHEMBL44632 0.83 LMNA (0.36)
SCHEMBL44454 0.83 CHEK2 (0.36) GSK3B
SCHEMBL44225 0.82 MAPT (0.50) TSHR
SCHEMBL44473 0.81 GRM5 (0.40)
SCHEMBL45706 0.81 SMPD1 (0.41) GSK3BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed