SCHEMBL4457095

SCHEMBL4457095

Nc1nc(N)c(Cc2cc(-c3ccc(F)cc3)no2)c(N2CCOCC2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.42
DRD4 P21917 5/20 0.42
DRD3 P35462 5/20 0.42
IGF1R P08069 2/20 0.42
NPC1 O15118 1/20 0.41
AR P10275 1/20 0.41
RAB9A P51151 1/20 0.41
NUDT1 P36639 1/20 0.40
RPS6KB1 P23443 1/20 0.40
KDM4E B2RXH2 3/20 0.39
TSHR P16473 3/20 0.39
ALDH1A1 P00352 2/20 0.39
NOS1 P29475 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIA1 P42261 1/20 0.38
CACNG2 Q9Y698 1/20 0.38
STK4 Q13043 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4469769 0.78 NUDT1 (0.46) IGF1RNUDT1KDM4ENOS1LMNA
SCHEMBL1791040 0.78 IGF1R (0.48) DRD2DRD4DRD3IGF1RHRH4
SCHEMBL4469774 0.76 NUDT1 (0.49) NUDT1KDM4EALDH1A1HSD17B10HPGD
SCHEMBL1787674 0.72 NOTUM (0.58) NPC1RAB9AKMT2ALMNAMAPT
SCHEMBL4114309 0.70 NOS1 (0.52) NPC1ARRAB9AKDM4ETSHR
SCHEMBL4363831 0.69 PRKDC (0.52) KDM4ETSHRALDH1A1HPGDGRIA1
SCHEMBL3983048 0.68 NOTUM (0.57) DRD2DRD4DRD3NPC1RAB9A
SCHEMBL4457078 0.68 IGF1R (0.41) IGF1RSTK4STK3HRH4HRH3
SCHEMBL4466081 0.67 DRD2 (0.41) DRD2DRD4DRD3IGF1RNPC1
SCHEMBL656484 0.67 NOS1 (0.44) NPC1ARRAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed