SCHEMBL4469774

SCHEMBL4469774

CCCc1cc(Cc2c(N)nc(N)nc2N2CCOCC2)on1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.49
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
MAP2K7 O14733 1/20 0.38
MBOAT4 Q96T53 3/20 0.36
PRKDC P78527 1/20 0.36
PIK3CA P42336 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
DHFR P00374 3/20 0.35
KDM4E B2RXH2 3/20 0.34
HPGD P15428 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 1/20 0.34
IKBKB O14920 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4462898 0.84 KDM4E (0.39) NUDT1PIK3CAMAPTDHFRKDM4E
SCHEMBL4469769 0.82 NUDT1 (0.46) NUDT1CRHBPCRHR2MAP2K7PRKDC
SCHEMBL4457095 0.76 DRD2 (0.42) NUDT1MAPTKDM4EHPGDALDH1A1
SCHEMBL4457348 0.72 HRH3 (0.35)
SCHEMBL4463994 0.72 IGF1R (0.31)
SCHEMBL4457078 0.70 IGF1R (0.41)
SCHEMBL17979717 0.68 NUDT1 (0.58) NUDT1CRHBPCRHR2MAP2K7PRKDC
SCHEMBL13650781 0.68 NUDT1 (0.61) NUDT1CRHBPCRHR2MAP2K7PRKDC
SCHEMBL4462891 0.67 IGF1R (0.43) PIK3CAMAPTKDM4EHPGDALDH1A1
SCHEMBL9643516 0.65 GAA (0.56) NUDT1CRHBPCRHR2MAP2K7PRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed