SCHEMBL446173

SCHEMBL446173

Fc1ccc(-c2ccnc(Cl)n2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.58
KMT2A Q03164 4/20 0.58
RAB9A P51151 2/20 0.58
NPC1 O15118 1/20 0.58
ATM Q13315 1/20 0.58
MAPT P10636 5/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
GAA P10253 1/20 0.47
KMO O15229 4/20 0.43
PIK3CA P42336 2/20 0.43
PIK3CG P48736 2/20 0.43
PIK3CB P42338 1/20 0.43
TRPV3 Q8NET8 1/20 0.42
TXN P10599 1/20 0.42
ALDH1A1 P00352 2/20 0.41
ALOX5 P09917 1/20 0.41
KDM4E B2RXH2 1/20 0.41
AR P10275 1/20 0.41
MAP4K4 O95819 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL441888 0.85 MAPT (0.59) MEN1KMT2ARAB9ANPC1MAPT
SCHEMBL3754047 0.82 MEN1 (0.56) MEN1KMT2ARAB9ANPC1ATM
SCHEMBL444442 0.82 KMT2A (0.56) MEN1KMT2ARAB9ANPC1ATM
SCHEMBL1667688 0.82 KMO (0.47) MEN1KMT2ARAB9ANPC1ATM
SCHEMBL28374207 0.82 KMO (0.41) MEN1KMT2ARAB9ANPC1ATM
SCHEMBL210678 0.82 MEN1 (0.66) MEN1KMT2ARAB9ANPC1ATM
SCHEMBL16161191 0.82 KMT2A (0.55) MEN1KMT2ARAB9AMAPTL3MBTL1
SCHEMBL443863 0.81 KIF11 (0.47) MEN1KMT2ARAB9ANPC1ATM
SCHEMBL31390937 0.81 MAPT (0.47) MEN1KMT2ARAB9ANPC1ATM
SCHEMBL445042 0.81 MEN1 (0.59) MEN1KMT2ARAB9AMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 70 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025067457-A1 HETEROCYCLIC FUSED RING COMPOUND, AND COMPOSITION AND USE THEREOF 深圳市塔吉瑞生物医药有限公司 2025-04-03 WO disclosed
US-20250026749-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GENZYME CORPORATION (US) 2025-01-23 US disclosed
US-12060349-B2 Glucosylceramide synthase inhibitors GENZYME CORPORATION (US) 2024-08-13 US disclosed
US-20230022534-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2023-01-26 US disclosed
EP-4098654-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS Genzyme Corporation (US) 2022-12-07 EP disclosed
CN-114533729-A Glucosylceramide synthase inhibitors 建新公司 2022-05-27 CN disclosed
US-20220073508-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GENZYME CORPORATION (US) 2022-03-10 US disclosed
EP-2895484-B1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GENZYME CORP (US) 2022-02-23 EP disclosed
CN-108864076-B Glucosylceramide synthase inhibitors 建新公司 2022-02-11 CN disclosed
US-11072611-B2 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders GALAPAGOS NV (BE) 2021-07-27 US disclosed
CN-101014587-A Substituted biaryl piperazinyl-pyridine analogues NEUROGEN CORP (US) 2007-08-08 CN disclosed
WO-2007016286-A1 SYNTHESIS OF 4/5-PYRIMIDINYLIMIDAZOLES VIA SEQUENTIAL FUNCTIONALIZATION OF 2,4-DICHLOROPYRIMIDINE JANSSEN PHARMACEUTICA N.V. (BE) 2007-02-08 WO disclosed
US-20070027319-A1 Synthesis of 4/5-pyrimidinylimidazoles via sequential functionalization of 2,4-dichloropyrimidine JANSSEN PHARMACEUTICA N.V. (BE) 2007-02-01 US disclosed
US-20060235004-A1 Pyrimidin-2-one compounds and their use as dopamine d3 receptor ligands ABBOT GMBH & CO. KG (DE) 2006-10-19 US disclosed
CN-1823057-A Biaryl piperazinyl-pyridine analogues NEUROGEN CORP (US) 2006-08-23 CN disclosed
EP-1601659-A1 PYRIMIDIN-2-ONE COMPOUNDS AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS Abbott GmbH & Co. KG (DE) 2005-12-07 EP disclosed
WO-2004080981-A1 PYRIMIDIN-2-ONE COMPOUNDS AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS ABBOTT GMBH & CO. KG (DE) 2004-09-23 WO disclosed
US-6440984-B1 PROTECTION FOR GROWING AND HARVESTED CROPS; CONTROLLING TOBACCO BUDWORMS AND SOUTHERN ARMYWORMS; PESTICIDES; INSECTICIDES; MITICIDES; ANTHELMINTICS BASF AKTIENGESELLSCHAFT (DE) 2002-08-27 US disclosed
US-6306866-B1 2-ALKOXY SUBSTITUTED PYRIMIDINE DERIVATIVES AMERICAN CYANAMID COMPANY 2001-10-23 US disclosed
US-6153619-A Aryl-substituted pyrimidines as insecticidal and acaricidal agents AMERICAN CYANAMID COMPANY (US) 2000-11-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11072611-B2 Compounds and pharmaceutical compositions thereof for the treatment of inflammatory disorders ENPP2, PRXL2A, TPX2 MEN1 3182/4885KMT2A 1634/4885RAB9A 1501/4885
US-20070027319-A1 Synthesis of 4/5-pyrimidinylimidazoles via sequential functionalization of 2,4-dichloropyrimidine DCK, DPYD, DTYMK MEN1 4120/4885KMT2A 1988/4885RAB9A 4275/4885
US-12060349-B2 Glucosylceramide synthase inhibitors GBA1, GBA2, GALC MEN1 1781/4885KMT2A 2942/4885RAB9A 490/4885
US-20250026749-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GBA1, GBA2, GAA MEN1 1532/4885KMT2A 2721/4885RAB9A 699/4885
US-20230022534-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS ENPP2, TPX2, PRXL2A MEN1 3384/4885KMT2A 1651/4885RAB9A 1170/4885
US-20060235004-A1 Pyrimidin-2-one compounds and their use as dopamine d3 receptor ligands ADRB3, DRD3, OPRL1 MEN1 4488/4885KMT2A 4190/4885RAB9A 3836/4885
US-20220073508-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GBA1, GBA2, GAA MEN1 1532/4885KMT2A 2721/4885RAB9A 699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.