SCHEMBL4463191

SCHEMBL4463191

Fc1ccc(C(Cl)(Cl)c2ccc(F)cc2F)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
KCNN4 O15554 1/20 0.42
CES2 O00748 2/20 0.38
CES1 P23141 2/20 0.38
CYP11B2 P19099 2/20 0.38
LMNA P02545 1/20 0.38
HSP90AA1 P07900 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP2C19 P33261 1/20 0.38
ADRA1A P35348 1/20 0.38
CYP51A1 Q16850 1/20 0.38
CA3 P07451 1/20 0.37
CA6 P23280 1/20 0.37
CA5A P35218 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
CA5B Q9Y2D0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11550172 0.85 ALDH1A1 (0.42) ALDH1A1KCNN4CES2CES1CYP11B2
SCHEMBL31433155 0.85 ALDH1A1 (0.42) ALDH1A1KCNN4CES2CES1CYP11B2
SCHEMBL4478794 0.80 CA3 (0.42) ALDH1A1KCNN4CES2CES1CA3
SCHEMBL4474477 0.78 CYP3A4 (0.43) ALDH1A1LMNACYP3A4CYP19A1CYP2C19
SCHEMBL22932517 0.78 KCNN4 (0.41) ALDH1A1KCNN4CES2CES1CYP11B2
SCHEMBL29490960 0.77 KIF11 (0.52) ALDH1A1KCNN4CYP11B2CYP11B1IDO1
SCHEMBL4084187 0.77 KIF11 (0.52) ALDH1A1KCNN4CYP11B2CYP11B1IDO1
SCHEMBL4468448 0.76 DGAT1 (0.39) ALDH1A1CYP11B2LMNACYP3A4CYP2C9
SCHEMBL441530 0.75 ALDH1A1 (0.42) ALDH1A1KCNN4CES2CES1CYP11B2
SCHEMBL22933206 0.75 KCNN4 (0.46) ALDH1A1KCNN4CES2CES1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576088-B2 Benzodioxole derivatives HOFFMAN-LA ROCHE INC. (US) 2009-08-18 US disclosed
EP-1532132-B1 NOVEL BENZODIOXOLES HOFFMANN LA ROCHE (CH) 2008-03-19 EP disclosed
US-20050143373-A1 Benzodioxole derivatives ALANINE ALEXANDER (FR) 2005-06-30 US disclosed
US-6900227-B2 Benzodioxole derivatives HOFFMANN-LA ROCHE INC. (US) 2005-05-31 US disclosed
EP-1532132-A1 NOVEL BENZODIOXOLES F.HOFFMANN-LA ROCHE AG (CH) 2005-05-25 EP disclosed
US-20040142922-A1 Benzodioxole derivatives HOFFMANN-LA ROCHE INC. 2004-07-22 US disclosed
WO-2004013120-A1 NOVEL BENZODIOXOLES F. HOFFMANN-LA ROCHE AG (CH) 2004-02-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050143373-A1 Benzodioxole derivatives CNR2, CNR1, GPR119 ALDH1A1 607/4885KCNN4 1843/4885CES2 197/4885
US-20040142922-A1 Benzodioxole derivatives CNR1, CNR2, GPR119 ALDH1A1 299/4885KCNN4 1690/4885CES2 214/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.