SCHEMBL4465339

SCHEMBL4465339

CCc1ccc(C(=O)N(CC)CC)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.43
HSP90AA1 P07900 4/20 0.42
HSP90AB1 P08238 4/20 0.42
CES2 O00748 2/20 0.39
LMNA P02545 1/20 0.39
RECQL P46063 1/20 0.39
PDE4B Q07343 1/20 0.38
TSHR P16473 2/20 0.37
GAA P10253 2/20 0.37
MCOLN3 Q8TDD5 1/20 0.37
ESRRG P62508 1/20 0.36
HPGD P15428 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MAPK1 P28482 1/20 0.36
PDK2 Q15119 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29175212 0.83 KMT2A (0.49) MLYCDHSP90AA1HSP90AB1CES2LMNA
SCHEMBL20178562 0.82 ALDH1A1 (0.46) CES2TSHRESRRGHPGD
SCHEMBL4470608 0.82 GAA (0.49) MLYCDHSP90AA1HSP90AB1GAAMCOLN3
SCHEMBL23370109 0.81 CES2 (0.43) CES2ESRRG
SCHEMBL14010461 0.80 CES2 (0.42) HSP90AB1CES2LMNAESRRGMAPK1
SCHEMBL23370103 0.80 GPR52 (0.45) CES2LMNAESRRGPDK2
SCHEMBL4469757 0.80 HSP90AA1 (0.45) MLYCDHSP90AA1HSP90AB1TSHRHPGD
SCHEMBL7306129 0.79 EPHX2 (0.46) LMNAPDE4BTSHRGAAMCOLN3
SCHEMBL3558708 0.78 HCRTR1 (0.47) MLYCDHSP90AA1HSP90AB1PDE4BTSHR
SCHEMBL10309762 0.78 CFTR (0.49) CES2TSHRGAAESRRGHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7572805-B2 Pyrrolo(oxo)isoquinolines as 5HT ligands BRISTOL-MYERS SQUIBB COMPANY (US) 2009-08-11 US disclosed
US-20060014777-A1 Pyrrolo(oxo)isoquinolines as 5HT ligands BRISTOL-MYERS SQUIBB COMPANY 2006-01-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060014777-A1 Pyrrolo(oxo)isoquinolines as 5HT ligands HTR2B, OPRD1, HTR1B MLYCD 1280/4885HSP90AA1 4652/4885HSP90AB1 4404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.