SCHEMBL4472978

SCHEMBL4472978

Nc1ncc(-c2ccc(CCN3CCCCC3)cc2)c(N)n1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.56
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.45
MBTD1 Q05BQ5 1/20 0.45
L3MBTL3 Q96JM7 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
SLC6A3 Q01959 1/20 0.43
CYP2D6 P10635 1/20 0.43
DHFR P00374 2/20 0.43
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
MCHR1 Q99705 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL265809 0.81 LTA4H (0.55) HRH3
SCHEMBL1935597 0.77 DHFR (0.51) DHFR
SCHEMBL17907568 0.76 LMNA (0.54) DHFR
SCHEMBL14694265 0.76 DHFR (0.58) L3MBTL1DHFR
SCHEMBL264111 0.74 HRH3 (0.56) HRH3DHFR
SCHEMBL2237239 0.74 DHFR (0.54) HRH3DHFR
Hydrochloric Acid SCHEMBL1935888 0.72 DHFR (0.53) HRH3DHFR
SCHEMBL29157674 0.72 DHFR (0.57) DHFRMCHR1
SCHEMBL2761916 0.71 HRH3 (0.71) HRH3CYP1A2CYP3A4L3MBTL1MBTD1
SCHEMBL2762024 0.71 HRH3 (0.71) HRH3CYP1A2CYP3A4L3MBTL1MBTD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed