Guanine

Guanine

SCHEMBL447498

Nc1cc[nH]c(=O)n1.Nc1nc2[nH]cnc2c(=O)[nH]1.O=P(O)(O)O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Guanine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
GLA P06280 1/20 0.43
PMP22 Q01453 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PNP P00491 5/20 0.38
HPRT1 P00492 7/20 0.36
AKR1B1 P15121 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Guanine SCHEMBL78999 0.94 DYRK1A (0.49) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL8470122 0.94 DYRK1A (0.49) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL76053 0.88 KDM4E (0.53) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL663745 0.88 KDM4E (0.53) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL13516878 0.85 KDM4E (0.44) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL1730016 0.85 DYRK1A (0.42) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL8471715 0.85 PNP (0.51) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL5372452 0.84 KDM4E (0.51) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL15948930 0.83 KDM4E (0.50) DYRK1AKDM4EALDH1A1LMNAGLA
Guanine SCHEMBL4007020 0.82 ATAD2 (0.41) DYRK1AKDM4EALDH1A1LMNAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 108 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118178636-A Immunogenic compositions and uses thereof 镁迪生医股份有限公司 2024-06-14 CN claimed
US-20230102739-A1 DETECTION OF EPIGENETIC MODIFICATIONS CAMBRIDGE EPIGENETIX LIMITED (GB) 2023-03-30 US claimed
EP-4013888-A1 METHODS AND KITS FOR INFERTILITY DIAGNOSTICS Washington State University (US) 2022-06-22 EP claimed
CN-114599800-A Method and kit for diagnosing infertility 华盛顿州立大学 2022-06-07 CN claimed
WO-2021030725-A1 METHODS AND KITS FOR INFERTILITY DIAGNOSTICS WASHINGTON STATE UNIVERSITY (US) 2021-02-18 WO claimed
US-10876163-B2 Detection and quality control of regulatory T cells through DNA-methylation analysis of the Foxp3 gene EPIONTIS GMBH (DE) 2020-12-29 US claimed
CN-112022836-A Preparation method of metal organic framework nano vaccine without refrigeration storage 山东大学 2020-12-04 CN claimed
CN-110997935-A Detection of epigenetic modifications 剑桥表现遗传学有限公司 2020-04-10 CN claimed
EP-3625365-A2 DETECTION OF EPIGENETIC MODIFICATIONS Cambridge Epigenetix Limited (GB) 2020-03-25 EP claimed
WO-2018211329-A2 DETECTION OF EPIGENETIC MODIFICATIONS CAMBRIDGE EPIGENETIX LIMITED (GB) 2018-11-22 WO claimed
EP-2729127-B1 METHODS FOR PRODUCING LIPOSOMES STATENS SERUMINSTITUT (DK) 2018-05-02 EP claimed
US-20140213475-A1 METHODS OF DIAGNOSING CANCER USING EPIGENETIC BIOMARKERS UNIVERSITY OF MASSACHUSETTS (US) 2014-07-31 US claimed
EP-2729127-A2 METHODS FOR PRODUCING LIPOSOMES Statens Serum Institut (DK) 2014-05-14 EP claimed
US-20140112979-A1 METHODS FOR PRODUCING LIPOSOMES STATENS SERUM INSTITUT (DK) 2014-04-24 US claimed
WO-2013010181-A2 METHODS OF DIAGNOSING CANCER USING EPIGENETIC BIOMARKERS UNIVERSITY OF MASSACHUSETTS (US) 2013-01-17 WO claimed
WO-2013004234-A2 METHODS FOR PRODUCING LIPOSOMES STATENS SERUM INSTITUT (DK) 2013-01-10 WO claimed
US-20240210288-A1 Representative Diagnostics VENTANA MED SYST INC (US) 2024-06-27 US disclosed
CN-118178636-A Immunogenic compositions and uses thereof 镁迪生医股份有限公司 2024-06-14 CN disclosed
EP-2200638-A1 A METHOD OF TRANSFECTION AND COMPOSITIONS THEREFOR THE UNIVERSITY OF MELBOURNE (AU) 2010-06-30 EP disclosed
WO-2009046498-A1 A METHOD OF TRANSFECTION AND COMPOSITIONS THEREFOR THE UNIVERSITY OF MELBOURNE (AU) 2009-04-16 WO disclosed