SCHEMBL44750

SCHEMBL44750

Cc1cn2cc(-c3cccc(CNCc4cccc(C#N)c4)c3)nc2s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.41
CYP2C19 P33261 4/20 0.41
HSD17B10 Q99714 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
SCN8A Q9UQD0 1/20 0.40
ALDH1A3 P47895 1/20 0.39
TGFBR1 P36897 3/20 0.39
MAPK14 Q16539 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
TP53 P04637 2/20 0.39
USP2 O75604 2/20 0.39
ALDH1A1 P00352 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44398 0.82 CHRM3 (0.52) TP53
SCHEMBL44636 0.77 TP53 (0.43) KDM4EMAPTHPGDPRMT6TP53
SCHEMBL44862 0.77 GAA (0.47) KDM4EMAPTHPGDTP53ALDH1A1
SCHEMBL44495 0.76 WDR5 (0.55) TSHRKDM4EMAPTHPGDALDH1A1
SCHEMBL45277 0.75 TP53 (0.49) CYP2C19HSD17B10CYP3A4KDM4EMAPT
SCHEMBL14207479 0.74 F2RL3 (0.53) CYP1A2CYP2C19KDM4EMAPTALDH1A3
SCHEMBL38543 0.74 WDR5 (0.45) CYP1A2CYP2C19HSD17B10MAPTHPGD
SCHEMBL44054 0.73 MAPT (0.53) KDM4EMAPTTP53LMNATHRB
SCHEMBL44267 0.73 ALDH1A3 (0.41) CYP1A2CYP2C19HSD17B10CYP3A4CYP2D6
SCHEMBL45795 0.73 CHRM3 (0.49) KDM4EMAPTTP53LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed