SCHEMBL447549

SCHEMBL447549

c1ccc(CON2CCCCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.47
LMNA P02545 1/20 0.46
LTA4H P09960 2/20 0.45
TSHR P16473 3/20 0.44
DHFR P00374 2/20 0.44
SLC6A3 Q01959 1/20 0.44
HRH3 Q9Y5N1 2/20 0.44
HPGD P15428 1/20 0.43
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9744353 1.00 SIGMAR1 (0.47) SIGMAR1LMNALTA4HTSHRDHFR
Bromide SCHEMBL28805308 0.98 SIGMAR1 (0.46) SIGMAR1LMNALTA4HTSHRDHFR
SCHEMBL2982806 0.98 TSHR (0.46) SIGMAR1LMNALTA4HTSHRDHFR
Hydrochloric Acid SCHEMBL2978407 0.96 LMNA (0.46) SIGMAR1LMNALTA4HTSHRDHFR
SCHEMBL15094370 0.94 TSHR (0.46) SIGMAR1LTA4HTSHRDHFRSLC6A3
SCHEMBL6620777 0.86 HRH3 (0.53) LTA4HHRH3
SCHEMBL10382845 0.81 ALDH1A1 (0.41) TSHRDHFRRAB9ANPC1
SCHEMBL28598923 0.80 TSHR (0.50) SIGMAR1LMNATSHRSLC6A3
SCHEMBL23279497 0.80 KMT2A (0.53) SIGMAR1LMNALTA4HTSHRHPGD
SCHEMBL20892082 0.80 MC4R (0.53) SIGMAR1LTA4HTSHRHRH3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119638614-A Recycling method of waste liquid generated in production of avibactam intermediate 德州宏海医药科技有限公司 2025-03-18 CN claimed
EP-0134124-B1 PIPERIDINE DERIVATIVES FORDONAL, S.A. (ES) 1987-10-28 EP claimed
EP-0134124-A1 Piperidine derivatives FORDONAL, S.A. (ES) 1985-03-13 EP claimed
EP-0015817-A1 Piperidine derivatives, process for their preparation and their use in therapeutical compositions METABIO-JOULLIE Société anonyme: (FR) 1980-09-17 EP claimed
CN-111423430-B Fluorescent probe and preparation method thereof 中山大学 2023-10-13 CN disclosed
CN-109689650-B Benzamide derivatives P2X7 receptor antagonists containing phenoxypiperidine or benzyloxypiperidine and thiazole 阿克萨姆股份公司 2022-11-25 CN disclosed
CN-109689650-B Benzamide derivatives P2X7 receptor antagonists containing phenoxypiperidine or benzyloxypiperidine and thiazole 阿克萨姆股份公司 2022-11-25 CN disclosed
CN-109689650-B Benzamide derivatives P2X7 receptor antagonists containing phenoxypiperidine or benzyloxypiperidine and thiazole 阿克萨姆股份公司 2022-11-25 CN disclosed
CN-114989169-A Preparation method of avibactam sodium 哈药集团技术中心 2022-09-02 CN disclosed
CN-114989169-A Preparation method of avibactam sodium 哈药集团技术中心 2022-09-02 CN disclosed
EP-3507287-B1 SUBSTITUTED N-[2-(4-PHENOXYPIPERIDIN-1-YL)-2-(1,3-THIAZOL-5-YL)ETHYL]BENZAMIDE AND N-[2-(4-BENZYLOXYPIPERIDIN-1-YL)-2-(1,3-THIAZOL-5-YL)ETHYL]BENZAMIDE DERIVATIVES P2X7 RECEPTOR ANTAGONISTS AXXAM SPA (IT) 2020-07-15 EP disclosed
US-10669267-B2 Substituted N-[2-(4-phenoxypiperidin-1-yl)-2-(1,3-thiazol-5-yl)ethyl]benzamide and N-[2-(4-benzyloxypiperidin-1-yl)-2-(1,3-thiazol-5-yl)ethyl]benzamide derivatives P2X7 receptor antagonists AXXAM S.P.A. (IT) 2020-06-02 US disclosed
CN-1039415-A New 1, the preparation method of 3-3-disubstituted piperidine derivatives PFIZER (GB) 1990-02-07 CN disclosed
EP-0134124-B1 PIPERIDINE DERIVATIVES FORDONAL, S.A. (ES) 1987-10-28 EP disclosed
US-4550116-A ANTIALLERGENS, CARDIOVASCULAR AND RESPIRATORY DISORDERS FORDONAL, S.A. (ES) 1985-10-29 US disclosed
EP-0077427-B1 PIPERIDINE DERIVATIVES, THEIR PREPARATION AND USE IN MEDICINE SYNTHELABO (FR) 1985-05-22 EP disclosed
EP-0134124-A1 Piperidine derivatives FORDONAL, S.A. (ES) 1985-03-13 EP disclosed
EP-0077427-A1 Piperidine derivatives, their preparation and use in medicine SYNTHELABO (FR) 1983-04-27 EP disclosed
EP-0015817-A1 Piperidine derivatives, process for their preparation and their use in therapeutical compositions METABIO-JOULLIE Société anonyme: (FR) 1980-09-17 EP disclosed
EP-0015817-A1 Piperidine derivatives, process for their preparation and their use in therapeutical compositions METABIO-JOULLIE Société anonyme: (FR) 1980-09-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10669267-B2 Substituted N-[2-(4-phenoxypiperidin-1-yl)-2-(1,3-thiazol-5-yl)ethyl]benzamide and N-[2-(4-benzyloxypiperidin-1-yl)-2-(1,3-thiazol-5-yl)ethyl]benzamide derivatives P2X7 receptor antagonists P2RX7, P2RX2, P2RX1 SIGMAR1 555/4885LMNA 1301/4885LTA4H 747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.