SCHEMBL448376

SCHEMBL448376

CNC(=S)N(c1ccccc1)N(C)S(=O)(=O)CC(=O)NN(C(=S)N(C)C)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 2/20 0.35
MMP3 P08254 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.31
HPGD P15428 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL446777 0.67 ALDH1A1 (0.36) LMNAL3MBTL1ALDH1A1SMN1; SMN2MEN1
SCHEMBL464694 0.64 ALDH1A1 (0.43) LMNAL3MBTL1ALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL10049995 0.62 HSP90AA1 (0.51) LMNAL3MBTL1ALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL13762631 0.60 MMP3 (0.57) LMNAALDH1A1MMP3SMN1; SMN2HSP90AA1
SCHEMBL6694830 0.59 LMNA (1.00) LMNAL3MBTL1ALDH1A1SMN1; SMN2MEN1
SCHEMBL10049989 0.58 HSP90AA1 (0.63) LMNAL3MBTL1ALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL9294461 0.58 ALDH1A1 (0.49) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL11810689 0.57 L3MBTL1 (0.67) LMNAL3MBTL1ALDH1A1SMN1; SMN2MEN1
SCHEMBL2810979 0.56 CA2 (0.39) LMNAL3MBTL1ALDH1A1SMN1; SMN2MEN1
SCHEMBL11684410 0.56 L3MBTL1 (0.54) LMNAL3MBTL1ALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8680100-B2 Sulfonylhydrazide compounds for treating proliferative disorders SYNTA PHARMACEUTICALS CORP. (US) 2014-03-25 US disclosed
US-20120065206-A1 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS SYNTA PHARMACEUTICALS CORP. (US) 2012-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120065206-A1 COMPOUNDS FOR TREATING PROLIFERATIVE DISORDERS PKD1, PKD2, PCNA LMNA 2213/4885L3MBTL1 4705/4885ALDH1A1 1351/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.